Inhibitors | Comment | Organism | Structure |
---|---|---|---|
elafin | 55% inhibition, oxidized with N-chlorosuccinimide: 10% inhibition | Homo sapiens | |
trappin | 80% inhibition, oxidized with N-chlorosuccinimide: 19% inhibition | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P24158 | - |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
neutrophil | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-p-nitroanilide + H2O | pH 7.4, 150 mM NaCl | Homo sapiens | ? | - |
? | |
methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester + H2O | pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine | Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PR3 | - |
Homo sapiens |
proteinase 3 | - |
Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00000012 | - |
elafin | methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine | Homo sapiens | |
0.00000018 | - |
trappin | methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine | Homo sapiens | |
0.000025 | - |
elafin, oxidized with myeloperoxidase | methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine | Homo sapiens | |
0.000029 | - |
elafin, oxidized with N-chlorosuccinimide | methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine | Homo sapiens | |
0.000035 | - |
trappin, oxidized with myeloperoxidase | methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine | Homo sapiens | |
0.00005 | - |
trappin, oxidized with N-chlorosuccinimide | methoxysuccinyl-lysyl-(2-picolinoyl)-Ala-Pro-Val-thiobenzylester as substrate, pH 7.4, 150 mM NaCl, 3 mM 4,4-dithiodipyridine | Homo sapiens |