Protein Variants | Comment | Organism |
---|---|---|
M156Q | mutation has no influence on the amidolytic and proteolytic activity of tissue factor bound enzyme, increased affinity for tissue factor | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
1.1 | - |
N-methylsulfonyl-D-Phe-Gly-Arg-p-nitroanilide | pH 8.0, 37°C, wild-type enzyme, addition of tissue factor | Homo sapiens | |
1.2 | - |
N-methylsulfonyl-D-Phe-Gly-Arg-p-nitroanilide | pH 8.0, 37°C, mutant enzyme M156Q, addition of tissue factor | Homo sapiens | |
5.3 | - |
N-methylsulfonyl-D-Phe-Gly-Arg-p-nitroanilide | pH 8.0, 37°C, mutant enzyme M156Q | Homo sapiens | |
7.6 | - |
N-methylsulfonyl-D-Phe-Gly-Arg-p-nitroanilide | pH 7.4, 37°C | Homo sapiens | |
61 | - |
Factor X | pH 7.4, 37°C, wild-type enzyme | Homo sapiens | |
68 | - |
Factor X | pH 7.4, 37°C, mutant enzyme | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
factor X + H2O | - |
Homo sapiens | ? | - |
? | |
N-methylsulfonyl-D-Phe-Gly-Arg-p-nitroanilide + H2O | i.e. chromozym t-PA | Homo sapiens | N-methylsulfonyl-D-Phe-Gly-Arg + p-nitroaniline | - |
? |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
8 | - |
Factor X | pH 7.4, 37°C, wild-type enzyme | Homo sapiens | |
10.2 | - |
Factor X | pH 7.4, 37°C, mutant enzyme | Homo sapiens | |
12.1 | - |
N-methylsulfonyl-D-Phe-Gly-Arg-p-nitroanilide | pH 8.0, 37°C, wild-type enzyme | Homo sapiens | |
24.6 | - |
N-methylsulfonyl-D-Phe-Gly-Arg-p-nitroanilide | pH 8.0, 37°C, mutant enzyme M156Q | Homo sapiens | |
49.1 | - |
N-methylsulfonyl-D-Phe-Gly-Arg-p-nitroanilide | pH 8.0, 37°C, wild-type enzyme, addition of tissue factor | Homo sapiens | |
49.8 | - |
N-methylsulfonyl-D-Phe-Gly-Arg-p-nitroanilide | pH 8.0, 37°C, mutant enzyme M156Q, addition of tissue factor | Homo sapiens |