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Literature summary for 3.4.21.122 extracted from

  • Meyer, D.; Sielaff, F.; Hammami, M.; Boettcher-Friebertshaeuser, E.; Garten, W.; Steinmetzer, T.
    Identification of the first synthetic inhibitors of the type II transmembrane serine protease TMPRSS2 suitable for inhibition of influenza virus activation (2013), Biochem. J., 452, 331-343 .
    View publication on PubMed
Search for more literature for 3.4.21.122

Cloned(Commentary)

Cloned (Comment) Organism
expression of the catalytic domain in Escherichia coli Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
1-[(2R)-4-(4-benzylpiperazin-1-yl)-4-oxo-2-[(phenylmethanesulfonyl)amino]butanoyl]-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
3-[(2S)-2-[(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-(4-[2-[(methylcarbamoyl)amino]ethyl]piperidin-1-yl)-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-2-[(2',4'-dimethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-(4-[2-[(methylcarbamoyl)amino]ethyl]piperidin-1-yl)-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-(2-aminoethyl)piperidin-1-yl]-2-[(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide treatment of cells with 10 microM inhibitor causes a 10fold and 100fold reduction in virus titres of A/Hamburg H1N1 and A/Aichi H3N2 respectively, at 24 h Homo sapiens
3-[(2S)-3-[4-[(cyclohexylcarbamoyl)amino]piperidin-1-yl]-2-[(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[(cyclohexylcarbamoyl)amino]piperidin-1-yl]-2-[(2',4'-dimethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2',3'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2',4'-dimethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2'-chloro-4'-ethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2'-chloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2'-fluoro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(3',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(3'-fluoro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(4'-chloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(4'-ethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(4'-fluoro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide
-
 Homo sapiens
4-[4-[([1-[3-carbamimidoyl-N-(2',3'-dichloro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide
-
 Homo sapiens
4-[4-[([1-[3-carbamimidoyl-N-(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide
-
 Homo sapiens
4-[4-[([1-[3-carbamimidoyl-N-(2',4'-dimethoxy[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide
-
 Homo sapiens
4-[4-[([1-[3-carbamimidoyl-N-(2'-chloro-4'-ethoxy[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide
-
 Homo sapiens
4-[4-[([1-[3-carbamimidoyl-N-(2'-fluoro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide
-
 Homo sapiens
4-[4-[([1-[3-carbamimidoyl-N-(3',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide
-
 Homo sapiens
4-[4-[([1-[3-carbamimidoyl-N-(3'-fluoro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide
-
 Homo sapiens
4-[4-[([1-[3-carbamimidoyl-N-(4'-fluoro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide
-
 Homo sapiens
5-oxo-N-(phenylmethanesulfonyl)-5-[4-(pyrimidin-2-yl)piperazin-1-yl]-D-norvalyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
5-[4-[(benzyloxy)carbonyl]piperazin-1-yl]-5-oxo-N-(phenylmethanesulfonyl)-D-norvalyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
benzyl 4-[(3R)-4-[(2S)-2-[[(4-carbamimidoylphenyl)methyl]carbamoyl]pyrrolidin-1-yl]-4-oxo-3-[(phenylmethanesulfonyl)amino]butanoyl]piperazine-1-carboxylate
-
 Homo sapiens
D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
D-homophenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-alaninamide
-
 Homo sapiens
D-homophenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
D-homotyrosinyl-N-[(4-carbamimidoylphenyl)methyl]-L-alaninamide
-
 Homo sapiens
D-phenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
methyl 1-[3-carbamimidoyl-N-(naphthalene-2-sulfonyl)-L-phenylalanyl]piperidine-4-carboxylate
-
 Homo sapiens
N-(3-[[(2S)-1-[4-(2-aminoethyl)piperidin-1-yl]-3-(3-carbamimidoylphenyl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-(4-[2-[(benzylcarbamoyl)amino]ethyl]piperidin-1-yl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-(4-[2-[(cyclohexylcarbamoyl)amino]ethyl]piperidin-1-yl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-(4-[2-[(ethylcarbamoyl)amino]ethyl]piperidin-1-yl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-(4-[2-[(methylcarbamoyl)amino]ethyl]piperidin-1-yl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-(4-[2-[(phenylcarbamoyl)amino]ethyl]piperidin-1-yl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[(benzylcarbamoyl)amino]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[(cyclohexylcarbamoyl)amino]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[(ethylcarbamoyl)amino]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[(methylcarbamoyl)amino]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[(phenylcarbamoyl)amino]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[2-(carbamoylamino)ethyl]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide
-
 Homo sapiens
N-(phenylmethanesulfonyl)-4-carbamimidoyl-D-phenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N-(phenylmethanesulfonyl)-4-cyano-D-phenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N-(phenylmethanesulfonyl)-D-alanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N-(phenylmethanesulfonyl)-D-alpha-aspartyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N-(phenylmethanesulfonyl)-D-cyclohexylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N-(phenylmethanesulfonyl)-D-leucyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N-(phenylmethanesulfonyl)-D-phenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N-(phenylmethanesulfonyl)-D-valyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N-(phenylmethanesulfonyl)-L-leucyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N-(phenylmethanesulfonyl)glycyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-(morpholin-4-yl)-4-oxo-2-[(phenylmethanesulfonyl)amino]butanoyl]-L-prolinamide
-
 Homo sapiens
N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-oxo-2-[(phenylmethanesulfonyl)amino]-4-(piperazin-1-yl)butanoyl]-L-prolinamide
-
 Homo sapiens
N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-oxo-2-[(phenylmethanesulfonyl)amino]-4-[4-(propan-2-yl)piperazin-1-yl]butanoyl]-L-prolinamide
-
 Homo sapiens
N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-oxo-2-[(phenylmethanesulfonyl)amino]-4-[4-(pyrimidin-2-yl)piperazin-1-yl]butanoyl]-L-prolinamide
-
 Homo sapiens
N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-[4-(2-hydroxyethyl)piperazin-1-yl]-4-oxo-2-[(phenylmethanesulfonyl)amino]butanoyl]-L-prolinamide
-
 Homo sapiens
N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-[4-(3,5-dimethylphenyl)piperazin-1-yl]-4-oxo-2-[(phenylmethanesulfonyl)amino]butanoyl]-L-prolinamide
-
 Homo sapiens
N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-[4-[3-(dimethylamino)propyl]piperazin-1-yl]-4-oxo-2-[(phenylmethanesulfonyl)amino]butanoyl]-L-prolinamide
-
 Homo sapiens
N-[3-([(2S)-3-(3-carbamimidoylphenyl)-1-[4-(carbamoylamino)piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl)phenyl]-beta-alaninamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-2-aminobutanoylamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-alaninamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-argininamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-isoleucinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-leucinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-norvalinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-phenylalaninamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-serinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-valinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]glycinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N-[[2-(aminomethyl)-5-chlorophenyl]methyl]-L-prolinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-arginyl-N6-[(benzyloxy)carbonyl]-N-[(4-carbamimidoylphenyl)methyl]-L-lysinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-homoarginyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-homophenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-D-lysyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-N-tert-butoxy-D-asparaginyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-N6-(benzyloxycarbonyl)-D-lysyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
N2-(phenylmethanesulfonyl)-O-(tert-butyl)-D-glutamyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide
-
 Homo sapiens
tert-butyl N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-alpha-asparaginate
-
 Homo sapiens

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
0.019
-
 CH3-SO2-D-cyclohexylalanine-Gly-Arg-4-nitroanilide pH 8.0, 23°C Homo sapiens
0.026
-
 CH3-SO2-D-cyclohexylglycine-Gly-Arg-4-nitroanilide pH 8.0, 23°C Homo sapiens
0.043
-
 CH3-SO2-D-Arg-Pro-Arg-7-amido-4-methylcoumarin pH 8.0, 23°C Homo sapiens
0.055
-
 CH3-O-CO-D-cyclohexylalanine-Gly-Arg-4-nitroanilide pH 8.0, 23°C Homo sapiens
0.058
-
 Boc-Phe-Ser-Arg-7-amido-4-methylcoumarin pH 8.0, 23°C Homo sapiens
0.059
-
 D-cyclohexylalanine-Gly-Arg-4-nitroanilide pH 8.0, 23°C Homo sapiens
0.065
-
 D-hexahydrotyrosine-Gly-Arg-4-nitroanilide pH 8.0, 23°C Homo sapiens
0.075
-
 Boc-Leu-GLy-Arg-7-amido-4-methylcoumarin pH 8.0, 23°C Homo sapiens
0.081
-
 Tos-Gly-Pro-Arg-7-amido-4-methylcoumarin pH 8.0, 23°C Homo sapiens
0.087
-
 D-Phe-Pro-Arg-7-amido-4-methylcoumarin pH 8.0, 23°C Homo sapiens
0.094
-
 Boc-Phe-Gly-Arg-7-amido-4-methylcoumarin pH 8.0, 23°C Homo sapiens
0.159
-
 Tos-Gly-Pro-Lys-7-amido-4-methylcoumarin pH 8.0, 23°C Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens O15393
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
Boc-Leu-GLy-Arg-7-amido-4-methylcoumarin + H2O
-
 Homo sapiens Boc-Leu-Gly-Arg + 7-amino-4-methylcoumarin
-
 ?
Boc-Phe-Gly-Arg-7-amido-4-methylcoumarin + H2O
-
 Homo sapiens Boc-Phe-Gly-Arg + 7-amino-4-methylcoumarin
-
 ?
Boc-Phe-Ser-Arg-7-amido-4-methylcoumarin + H2O
-
 Homo sapiens Boc-Phe-Ser-Arg + 7-amino-4-methylcoumarin
-
 ?
CH3-O-CO-D-cyclohexylalanine-Gly-Arg-4-nitroanilide + H2O 58% of the activtiy with CH3-SO2-D-Arg-Gly-Arg-4-nitroanilide Homo sapiens CH3-O-CO-D-cyclohexylalanine-Gly-Arg + 4-nitroaniline
-
 ?
CH3-SO2-D-Arg-Gly-Arg-4-nitroanilide + H2O
-
 Homo sapiens CH3-SO2-D-Arg-Gly-Arg + 4-nitroaniline
-
 ?
CH3-SO2-D-Arg-Pro-Arg-7-amido-4-methylcoumarin + H2O
-
 Homo sapiens CH3-SO2-D-Arg-Pro-Arg + 7-amino-4-methylcoumarin
-
 ?
CH3-SO2-D-cyclohexylalanine-Gly-Arg-4-nitroanilide + H2O 54% of the activtiy with CH3-SO2-D-Arg-Gly-Arg-4-nitroanilide Homo sapiens CH3-SO2-D-cyclohexylalanine-Gly-Arg-4-nitroaniline
-
 ?
CH3-SO2-D-cyclohexylglycine-Gly-Arg-4-nitroanilide + H2O 70% of the activtiy with CH3-SO2-D-Arg-Gly-Arg-4-nitroanilide Homo sapiens CH3-SO2-D-cyclohexylglycine-Gly-Arg + 4-nitroaniline
-
 ?
D-cyclohexylalanine-Gly-Arg-4-nitroanilide + H2O
-
 Homo sapiens D-cyclohexylalanine-Gly-Arg + 4-nitroaniline
-
 ?
D-hexahydrotyrosine-Gly-Arg-4-nitroanilide + H2O 87% of the activtiy with CH3-SO2-D-Arg-Gly-Arg-4-nitroanilide Homo sapiens D-hexahydrotyrosine-Gly-Arg + 4-nitroaniline
-
 ?
D-Phe-Pro-Arg-7-amido-4-methylcoumarin + H2O
-
 Homo sapiens D-Phe-Pro-Arg + 7-amino-4-methylcoumarin
-
 ?
Tos-Gly-Pro-Arg-7-amido-4-methylcoumarin + H2O
-
 Homo sapiens Tos-Gly-Pro-Arg + 7-amino-4-methylcoumarin
-
 ?
Tos-Gly-Pro-Lys-7-amido-4-methylcoumarin + H2O
-
 Homo sapiens Tos-Gly-Pro-Lys + 7-amino-4-methylcoumarin
-
 ?

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.0000009
-
 3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000001
-
 3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2',4'-dimethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.0000027
-
 3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2',3'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000003
-
 3-[(2S)-3-[4-[(cyclohexylcarbamoyl)amino]piperidin-1-yl]-2-[(2',4'-dimethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000004
-
 4-[4-[([1-[3-carbamimidoyl-N-(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.0000045
-
 4-[4-[([1-[3-carbamimidoyl-N-(2',4'-dimethoxy[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.0000048
-
 3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(4'-ethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000005
-
 3-[(2S)-3-[4-[(cyclohexylcarbamoyl)amino]piperidin-1-yl]-2-[(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.0000054
-
 3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(4'-chloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000006
-
 N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[(cyclohexylcarbamoyl)amino]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000007
-
 N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-(4-[2-[(phenylcarbamoyl)amino]ethyl]piperidin-1-yl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.0000073
-
 3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(4'-chloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.0000078
-
 3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2'-chloro-4'-ethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000008
-
 N-(3-[[(2S)-1-[4-(2-aminoethyl)piperidin-1-yl]-3-(3-carbamimidoylphenyl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00001
-
 N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-(4-[2-[(methylcarbamoyl)amino]ethyl]piperidin-1-yl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000011
-
 N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-(4-[2-[(ethylcarbamoyl)amino]ethyl]piperidin-1-yl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000011
-
 3-[(2S)-2-[(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-(4-[2-[(methylcarbamoyl)amino]ethyl]piperidin-1-yl)-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000013
-
 3-[(2S)-2-[(2',4'-dimethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-(4-[2-[(methylcarbamoyl)amino]ethyl]piperidin-1-yl)-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000016
-
 N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[2-(carbamoylamino)ethyl]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000017
-
 N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[(phenylcarbamoyl)amino]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000017
-
 4-[4-[([1-[3-carbamimidoyl-N-(2'-chloro-4'-ethoxy[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000018
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000018
-
 N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-(4-[2-[(benzylcarbamoyl)amino]ethyl]piperidin-1-yl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000019
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000019
-
 N2-(phenylmethanesulfonyl)-N-tert-butoxy-D-asparaginyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000019
-
 4-[4-[([1-[3-carbamimidoyl-N-(2',3'-dichloro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00002
-
 N2-(phenylmethanesulfonyl)-D-lysyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00002
-
 D-homotyrosinyl-N-[(4-carbamimidoylphenyl)methyl]-L-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000021
-
 N2-(phenylmethanesulfonyl)-D-homoarginyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000021
-
 N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[(benzylcarbamoyl)amino]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000022
-
 N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-(4-[2-[(cyclohexylcarbamoyl)amino]ethyl]piperidin-1-yl)-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000025
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-argininamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000028
-
 3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(4'-fluoro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000028
-
 3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2'-fluoro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000036
-
 4-[4-[([1-[3-carbamimidoyl-N-(3',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00004
-
 4-[4-[([1-[3-carbamimidoyl-N-(2'-fluoro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000045
-
 N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-oxo-2-[(phenylmethanesulfonyl)amino]-4-(piperazin-1-yl)butanoyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00005
-
 N2-(phenylmethanesulfonyl)-D-homophenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00005
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N6-[(benzyloxy)carbonyl]-N-[(4-carbamimidoylphenyl)methyl]-L-lysinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000052
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-2-aminobutanoylamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00006
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[[2-(aminomethyl)-5-chlorophenyl]methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000068
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-norvalinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000068
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]glycinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000072
-
 3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(3'-fluoro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000072
-
 4-[4-[([1-[3-carbamimidoyl-N-(4'-fluoro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000074
-
 N-[3-([(2S)-3-(3-carbamimidoylphenyl)-1-[4-(carbamoylamino)piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl)phenyl]-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000081
-
 N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[(methylcarbamoyl)amino]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000089
-
 3-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(3',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00009
-
 D-homophenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000101
-
 N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-(morpholin-4-yl)-4-oxo-2-[(phenylmethanesulfonyl)amino]butanoyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000111
-
 N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-[4-(3,5-dimethylphenyl)piperazin-1-yl]-4-oxo-2-[(phenylmethanesulfonyl)amino]butanoyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000123
-
 N-(phenylmethanesulfonyl)-4-carbamimidoyl-D-phenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000143
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-serinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000166
-
 N-(phenylmethanesulfonyl)-D-phenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00018
-
 D-homophenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00018
-
 methyl 1-[3-carbamimidoyl-N-(naphthalene-2-sulfonyl)-L-phenylalanyl]piperidine-4-carboxylate 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000184
-
 N2-(phenylmethanesulfonyl)-N6-(benzyloxycarbonyl)-D-lysyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000207
-
 4-[4-[([1-[3-carbamimidoyl-N-(3'-fluoro[1,1'-biphenyl]-3-sulfonyl)-L-phenylalanyl]piperidin-4-yl]carbamoyl)amino]cyclohexyl]-N-methylbutanamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00021
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-phenylalaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00022
-
 D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00023
-
 N2-(phenylmethanesulfonyl)-O-(tert-butyl)-D-glutamyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000244
-
 N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-oxo-2-[(phenylmethanesulfonyl)amino]-4-[4-(propan-2-yl)piperazin-1-yl]butanoyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000248
-
 N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-[4-[3-(dimethylamino)propyl]piperazin-1-yl]-4-oxo-2-[(phenylmethanesulfonyl)amino]butanoyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000272
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-leucinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000322
-
 N-(phenylmethanesulfonyl)-D-valyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000335
-
 N-(phenylmethanesulfonyl)-D-cyclohexylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000363
-
 1-[(2R)-4-(4-benzylpiperazin-1-yl)-4-oxo-2-[(phenylmethanesulfonyl)amino]butanoyl]-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000393
-
 N-(phenylmethanesulfonyl)-D-leucyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000409
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-valinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.00041
-
 N-(3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[(ethylcarbamoyl)amino]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl)-beta-alaninamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000417
-
 N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-[4-(2-hydroxyethyl)piperazin-1-yl]-4-oxo-2-[(phenylmethanesulfonyl)amino]butanoyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000499
-
 N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-isoleucinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000624
-
 benzyl 4-[(3R)-4-[(2S)-2-[[(4-carbamimidoylphenyl)methyl]carbamoyl]pyrrolidin-1-yl]-4-oxo-3-[(phenylmethanesulfonyl)amino]butanoyl]piperazine-1-carboxylate 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000706
-
 N-(phenylmethanesulfonyl)-4-cyano-D-phenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000738
-
 tert-butyl N2-(phenylmethanesulfonyl)-D-arginyl-N-[(4-carbamimidoylphenyl)methyl]-L-alpha-asparaginate 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000821
-
 5-oxo-N-(phenylmethanesulfonyl)-5-[4-(pyrimidin-2-yl)piperazin-1-yl]-D-norvalyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.000838
-
 N-[(4-carbamimidoylphenyl)methyl]-1-[(2R)-4-oxo-2-[(phenylmethanesulfonyl)amino]-4-[4-(pyrimidin-2-yl)piperazin-1-yl]butanoyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.001222
-
 5-[4-[(benzyloxy)carbonyl]piperazin-1-yl]-5-oxo-N-(phenylmethanesulfonyl)-D-norvalyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.001633
-
 N-(phenylmethanesulfonyl)glycyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.001637
-
 N-(phenylmethanesulfonyl)-D-alanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.0029
-
 D-phenylalanyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens
0.007344
-
 N-(phenylmethanesulfonyl)-D-alpha-aspartyl-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide 50 mM Tris/HCl buffer, pH 8.0, 22°C Homo sapiens