EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
4.1.1.15 | 0.0002 |
- |
3,3'-(4H-1,2,4-triazole-3,5-diyl)bis(4-nitro-1,2,5-oxadiazole) |
pH 8.0, 37°C, recombinant enzyme |
727626 |
4.1.1.15 | 0.0004 |
- |
3,3'-(4H-1,2,4-triazole-3,5-diyl)bis(4-nitro-1,2,5-oxadiazole) |
pH 8.0, 37°C, recombinant enzyme |
727626 |
4.1.1.15 | 0.0004 |
- |
carboxymethoxylamine |
pH 8.0, 37°C, recombinant enzyme |
727626 |
4.1.1.15 | 0.0005 |
- |
carboxymethoxylamine |
pH 8.0, 37°C, recombinant enzyme |
727626 |
4.1.1.15 | 0.001 |
- |
carboxymethoxylamine |
pH 8.0, 37°C, recombinant enzyme |
727626 |
4.1.1.15 | 0.001 |
- |
methyl 2-amino-3-oxo-3H-phenothiazine-1-carboxylate |
pH 8.0, 37°C, recombinant enzyme |
727626 |
4.1.1.15 | 0.001 |
- |
N-[4,7-dioxo-6-(phenylamino)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide |
pH 8.0, 37°C, recombinant enzyme |
727626 |
4.1.1.15 | 0.0011 |
- |
N-[4,7-dioxo-6-(phenylamino)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide |
pH 8.0, 37°C, recombinant enzyme |
727626 |
4.1.1.15 | 0.0012 |
- |
N-[4,7-dioxo-6-(phenylamino)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide |
pH 8.0, 37°C, recombinant enzyme |
727626 |
4.1.1.15 | 0.0013 |
- |
N-[4,7-dioxo-6-(piperidin-1-yl)-4,7-dihydro-2,1,3-benzoxadiazol-5-yl]acetamide |
pH 8.0, 37°C, recombinant enzyme |
727626 |