EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    3.1.1.4 | -999 |
- |
more |
- |
681300 |
| 3.1.1.4 | -999 |
- |
more |
IC50 values of diverse isozymes, overview |
693563 |
| 3.1.1.4 | -999 |
- |
more |
inhibition of cPLA2a activity in the isolated enzyme assay and in the cellular assay, overview |
691215 |
| 3.1.1.4 | 0.000005 |
- |
1-[2-oxo-3-(4-phenoxyphenoxy)propyl]-1H-indazole-5-carboxylic acid |
37°C, pH 8.0, substrate 1-stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine |
754278 |
| 3.1.1.4 | 0.000005 |
- |
1-[3-(4-octylphenoxy)-2-oxopropyl]indazole-5-carboxylic acid |
- |
707663 |
| 3.1.1.4 | 0.000006 |
- |
2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-6,7-benzoindol-4-yloxy)acetic acid |
isozyme sPLA2 group IIX |
693563 |
| 3.1.1.4 | 0.000007 |
- |
2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-6,7-benzoindol-4-yloxy)acetic acid |
isozymes sPLA2 group IIE and IID |
693563 |
| 3.1.1.4 | 0.000007 |
- |
2-([3-[amino(oxo)acetyl]-1-benzyl-2-(2-methylpropyl)-1H-indol-4-yl]oxy)-N-(methylsulfonyl)propanamide |
isozyme sPLA2 group IIX |
693563 |
| 3.1.1.4 | 0.000007 |
- |
2-([3-[amino(oxo)acetyl]-1-benzyl-2-ethyl-1H-indol-4-yl]oxy)-N-(phenylsulfonyl)acetamide |
isozyme sPLA2 group IIE |
693563 |
| 3.1.1.4 | 0.000009 |
- |
2-[1-benzyl-4-(2-oxopropoxy)-2-propyl-1H-indol-3-yl]-2-oxoacetamide |
isozyme sPLA2 group IIE |
693563 |
