EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.13.11.34 | -999 |
- |
more |
enzyme inhibition in presence of inhibitor and glutathione peroxidase, overview |
684399 |
1.13.11.34 | -999 |
- |
more |
inhibitory activity in polymorphonuclear leukocytes, overview |
689841 |
1.13.11.34 | 0.000003 |
- |
3-[[3-fluoro-5-(4-methoxytetrahydro-2H-pyran-4-yl)phenoxy]methyl]-1-[4-(methylsulfonyl)phenyl]-5-phenyl-1H-pyrazole |
in 100 mM phosphate buffer, pH 6.3, 25°C |
711397 |
1.13.11.34 | 0.000009 |
- |
7-([3-fluoro-5-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenyl]sulfanyl)-4-furan-3-yl-2H-chromen-2-one |
IC50: 9 nM |
672591 |
1.13.11.34 | 0.00001 |
- |
4-methoxy-4-[3-(naphthalen-2-ylmethoxy)phenyl]tetrahydro-2H-pyran |
in 100 mM phosphate buffer, pH 6.3, 25°C |
711397 |
1.13.11.34 | 0.000014 |
- |
7-[[3-(4-methoxytetrahydro-2H-pyran-4-yl)benzyl]oxy]-4-phenylnaphtho[2,3-c]furan-1(3H)-one |
in 100 mM phosphate buffer, pH 6.3, 25°C |
711397 |
1.13.11.34 | 0.000015 |
- |
4-(furan-3-yl)-7-[[6-(4-hydroxytetrahydro-2H-pyran-4-yl)pyridin-2-yl]methoxy]naphthalene-2-carbonitrile |
in 100 mM phosphate buffer, pH 6.3, 25°C |
711397 |
1.13.11.34 | 0.000015 |
- |
7-[[3-(1-ethyl-1-hydroxypropyl)-5-fluorophenoxy]methyl]-4-furan-3-yl-2H-chromen-2-one |
IC50: 15 nM |
672591 |
1.13.11.34 | 0.000016 |
- |
1-(4-chlorobenzyl)-2-[2,2-dimethyl-3-(1H-tetrazol-5-yl)propyl]-4-methyl-6-[2-(5-phenylpyridin-2-yl)ethyl]-2,2a,4,5-tetrahydro-1H-thiopyrano[2,3,4-cd]indole |
in 100 mM phosphate buffer, pH 6.3, 25°C |
711397 |
1.13.11.34 | 0.00002 |
- |
L-697,198 |
IC50: 0.00002 mM |
439464 |