EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
    3.6.1.1 | -999 |
- |
more |
inhibition kinetics |
685299 |
| 3.6.1.1 | 0.0028 |
- |
fluoride |
pH 7.4, 25°C, with 0.05 mM Mn2+ |
688341 |
| 3.6.1.1 | 0.011 |
- |
4-(azepan-1-yl)-N,N-dibutyl-6-[1-(2-phenylethyl)-1H-pyrrol-2-yl]-1,3,5-triazin-2-amine |
recombinant enzyme, pH 7.5, 37°C |
755676 |
| 3.6.1.1 | 0.012 |
- |
fluoride |
pH 7.2, 25°C, wild-type enzyme, kinetics |
687549 |
| 3.6.1.1 | 0.025 |
- |
p-chloromercuriphenyl sulfonate |
- |
209819 |
| 3.6.1.1 | 0.033 |
- |
hydroxymethylbisphosphonate |
pH 7.2 |
654598 |
| 3.6.1.1 | 0.0358 |
- |
fluoride |
pH 7.4, 25°C, with 5 mM Mn2+ |
688341 |
| 3.6.1.1 | 0.33 |
- |
Methylenediphosphonate |
pH 7.5, 25°C, wild-type mutant |
685299 |
| 3.6.1.1 | 0.42 |
- |
more |
pH 7.2, 37°C, fluoride inhibition kinetics |
684535 |
