Cloned (Comment) | Organism |
---|---|
expression in Pichia pastoris | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
alpha2-antiplasmin | 50% inhibition at 0.8 microM in 0.6 min | Homo sapiens | |
antithrombin III | 50% inhibition at 0.8 microM in 6 min | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.02 | - |
Boc-Val-Pro-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.15 | - |
Boc-Leu-GLy-Arg-7-amido-4-methylcoumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.19 | - |
Boc-Phe-Ser-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.31 | - |
Z-Gly-Gly-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.48 | - |
Boc-Leu-Arg-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.57 | - |
Boc-Gln-Gly-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.61 | - |
Boc-Gln-Ala-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.64 | - |
Boc-Val-Leu-Lys-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
1.01 | - |
Boc-Leu-Lys-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
1.41 | - |
Boc-Gln-Arg-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
1.69 | - |
Tos-Gly-Pro-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
1.77 | - |
H-Pro-Phe-Ser-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
26000 | - |
calculated from sequence | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Posttranslational Modification | Comment | Organism |
---|---|---|
glycoprotein | - |
Homo sapiens |
Purification (Comment) | Organism |
---|---|
two chromatography steps, 95% purity | Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Boc-Gln-Ala-Arg-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | Boc-Gln-Ala-Arg + 7-amino-4-methyl-coumarin | - |
? | |
Boc-Gln-Arg-Arg-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | Boc-Gln-Arg-Arg + 7-amino-4-methyl-coumarin | - |
? | |
Boc-Gln-Gly-Arg-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | Boc-Gln-Gly-Arg + 7-amino-4-methyl-coumarin | - |
? | |
Boc-Leu-Arg-Arg-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | Boc-Leu-Arg-Arg + 7-amino-4-methyl-coumarin | - |
? | |
Boc-Leu-GLy-Arg-7-amido-4-methylcoumarin + H2O | - |
Homo sapiens | Boc-Leu-Gly-Arg + 7-amino-4-methylcoumarin | - |
? | |
Boc-Leu-Lys-Arg-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | Boc-Leu-Lys-Arg + 7-amino-4-methyl-coumarin | - |
? | |
Boc-Phe-Ser-Arg-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | Boc-Phe-Ser-Arg + 7-amino-4-methyl-coumarin | - |
? | |
Boc-Val-Leu-Lys-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | Boc-Val-Leu-Lys + 7-amino-4-methyl-coumarin | - |
? | |
Boc-Val-Pro-Arg-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | Boc-Val-Pro-Arg + 7-amino-4-methyl-coumarin | - |
? | |
casein + H2O | - |
Homo sapiens | ? | - |
? | |
fibrinogen Aalpha chain + H2O | cleavage after Arg348 and Arg407 | Homo sapiens | ? | - |
? | |
fibrinogen Bbeta chain + H2O | cleavage after Lys53 and Arg14 | Homo sapiens | ? | - |
? | |
Gelatin + H2O | - |
Homo sapiens | ? | - |
? | |
H-Pro-Phe-Ser-Arg-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | H-Pro-Phe-Ser-Arg + 7-amino-4-methyl-coumarin | - |
? | |
kininogen + H2O | cleavage after Arg222, Arg252 and Arg374 | Homo sapiens | ? | - |
? | |
plasminogen + H2O | cleavage after Lys77 andA rg529 | Homo sapiens | ? | - |
? | |
Pro-Phe-Ser-Arg-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | Pro-Phe-Ser-Arg + 7-amino-4-methyl-coumarin | - |
? | |
Tos-Gly-Pro-Arg-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | Tos-Gly-Pro-Arg + 7-amino-4-methyl-coumarin | - |
? | |
Vitronectin + H2O | cleavage after Arg8 | Homo sapiens | ? | - |
? | |
Z-Gly-Gly-Arg-7-amido-4-methyl-coumarin + H2O | - |
Homo sapiens | Z-Gly-Gly-Arg + 7-amino-4-methyl-coumarin | - |
? |
Synonyms | Comment | Organism |
---|---|---|
hK5 | - |
Homo sapiens |
human kallikrein 5 | - |
Homo sapiens |
KLK5 | - |
Homo sapiens |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.04 | - |
Z-Gly-Gly-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.07 | - |
Boc-Leu-GLy-Arg-7-amido-4-methylcoumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.08 | - |
Boc-Val-Leu-Lys-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.18 | - |
Boc-Gln-Gly-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.31 | - |
Boc-Leu-Arg-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.35 | - |
Tos-Gly-Pro-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.41 | - |
Boc-Gln-Arg-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.47 | - |
H-Pro-Phe-Ser-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
0.82 | - |
Boc-Leu-Lys-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
1.78 | - |
Boc-Gln-Ala-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
2.83 | - |
Boc-Phe-Ser-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens | |
3.28 | - |
Boc-Val-Pro-Arg-7-amido-4-methyl-coumarin | 100 mM phosphate, 0.01% Tween 20, pH 8.0, 37°C | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
8 | - |
- |
Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00107 | - |
alpha2-antiplasmin | - |
Homo sapiens | |
0.0091 | - |
antithrombin III | - |
Homo sapiens |