EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
7.5.2.6 | 0.000005 |
- |
(2E)-3-[1-cyclopropyl-7-[(1S)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]naphthalen-2-yl]prop-2-enoic acid |
pH 7.5, 37°C, recombinant detagged enzyme |
751693 |
7.5.2.6 | 0.000018 |
- |
(2E)-3-[6-[1-(2-chloro-6-cyclopropylphenyl)ethoxy]-4-cyclopropylquinolin-3-yl]prop-2-enoic acid |
pH 7.5, 37°C, recombinant detagged enzyme |
751693 |
7.5.2.6 | 0.48 |
- |
leupeptin |
pH 7.5, 37°C, recombinant His-tagged enzyme |
698746 |
7.5.2.6 | 0.5 |
- |
vinblastin |
above, pH 7.5, 37°C, recombinant His-tagged enzyme |
698746 |
7.5.2.6 | 1.25 |
- |
AMP-PCP |
pH 7.5, 37°C, recombinant His-tagged protein |
698746 |