EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   7.2.2.10 | 0.00016 |
- |
cyclopiazonic acid |
in 1 mM EGTA, 130 mM NaCl, 3 mM MgCl2, at 37°C |
695867 |
| 7.2.2.10 | 0.0004 |
- |
cyclopiazonic acid |
at pH 7.5 and 25°C |
733830 |
| 7.2.2.10 | 0.0004 |
- |
palytoxin |
in 20 mM MOPS, pH 7.0, 80 mM KC1, 5 mM MgCl2, 0.5 mM EGTA, 0.55 mM CaC12, at 25°C |
695863 |
| 7.2.2.10 | 0.000635 |
- |
thapsigargin |
recombinant enzyme expressed in Saccharomyces cerevisiae strain HI227, in 1 mM EGTA, 130 mM NaCl, 3 mM MgCl2, at 37°C |
695867 |
| 7.2.2.10 | 0.0008 |
- |
N-((3-chlorophenyl)(4-((4-(7-chloroquinolin-4-yl)piperazin-1-yl)methyl)phenyl)methyl)-7-chloro-4-aminoquinoline |
in 20 mM MOPS, pH 6.8, 80 mM KCl, 3 mM MgCl2, 0.002 mM A23187, 5 mM sodium azide, and 2 mM EGTA, or 0.2 mM EGTA plus 0.2 mM CaCl2, at 37°C |
719980 |
| 7.2.2.10 | 0.00095 |
- |
thapsigargin |
recombinant enzyme expressed in Saccharomyces cerevisiae strain K616, in 1 mM EGTA, 130 mM NaCl, 3 mM MgCl2, at 37°C |
695867 |
| 7.2.2.10 | 0.001 |
- |
2,3-bis[(2-hydroxyethyl)sulfanyl]naphthalene-1,4-dione |
at pH 7.5 and 25°C |
733830 |
| 7.2.2.10 | 0.001 |
- |
2-phenyl-1,2-benzoselenazol-3(2H)-one |
at pH 7.5 and 25°C |
733830 |
| 7.2.2.10 | 0.0011 |
- |
4,5-dimethyl-2-([[5-methyl-2-(propan-2-yl)phenoxy]acetyl]amino)thiophene-3-carboxamide |
at pH 7.5 and 25°C |
733830 |
| 7.2.2.10 | 0.0012 |
- |
methyl [(4-tert-butylbenzoyl)amino]acetate |
at pH 7.5 and 25°C |
733830 |
