EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
6.1.1.2 | 0.000002 |
- |
indolmycin |
pH 8.0, 37°C, recombinant enzyme |
745352 |
6.1.1.2 | 0.0151 |
- |
3-[(4-[[4-oxo-2-(phenylimino)-1,3-thiazolidin-5-ylidene]methyl]phenoxy) methyl]benzoic acid |
pH 8.0, 25°C, assay method b |
674218 |
6.1.1.2 | 0.0183 |
- |
3-[(4-[[4-oxo-2-(phenylimino)-1,3-thiazolidin-5-ylidene]methyl]phenoxy) methyl]benzoic acid |
pH 8.0, 25°C, assay method a |
674218 |
6.1.1.2 | 0.0187 |
- |
2-[5-[(6-(ethoxycarbonyl)-5-(4-fluorophenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-2(3H)-ylidene)methyl]-2-furyl]benzoic acid |
pH 8.0, 25°C, assay method b |
674218 |
6.1.1.2 | 0.0228 |
- |
2-[5-[(6-(ethoxycarbonyl)-5-(4-fluorophenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-2(3H)-ylidene)methyl]-2-furyl]benzoic acid |
pH 8.0, 25°C, assay method a |
674218 |
6.1.1.2 | 0.0352 |
- |
3-[[([[2-(4-chlorophenyl)-4-quinolinyl]carbonyl]amino)carbothioyl]amino]benzoic acid |
pH 8.0, 25°C, assay method b |
674218 |
6.1.1.2 | 0.0422 |
- |
3-[[([[2-(4-chlorophenyl)-4-quinolinyl]carbonyl]amino)carbothioyl]amino]benzoic acid |
pH 8.0, 25°C, assay method a |
674218 |