EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
5.3.99.3 | 0.0000007 |
- |
2-[6-chloro-9-(3-hydroxy-3-methylbutyl)-1H-phenanthro[9,10-d]imidazol-2-yl]benzene-1,3-dicarbonitrile |
- |
693551 |
5.3.99.3 | 0.0000008 |
- |
biarylimidazole |
- |
693551 |
5.3.99.3 | 0.0000009 |
- |
2-(difluoromethyl)-5-[(2-methylpropanamido)methyl]-N-[4-methyl-5-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]pyridine-3-carboxamide |
at pH 7.0 and 25°C |
748368 |
5.3.99.3 | 0.0000009 |
- |
2-(difluoromethyl)-5-[(2-methylpropanamido)methyl]-N-[5-methyl-4-[4-(trifluoromethyl)phenyl]-1H-imidazol-2-yl]pyridine-3-carboxamide |
pH and temperature not specified in the publication |
747282 |
5.3.99.3 | 0.0000009 |
- |
2-[6-(2-cyclopropylethoxy)-9-(3-hydroxy-3-methylbutyl)-1H-phenanthro[9,10-d]imidazol-2-yl]benzene-1,3-dicarbonitrile |
- |
693551 |
5.3.99.3 | 0.0000009 |
- |
2-[6-bromo-9-(3-hydroxy-3-methylbut-1-yn-1-yl)-1H-phenanthro[9,10-d]imidazol-2-yl]benzene-1,3-dicarbonitrile |
- |
693551 |
5.3.99.3 | 0.0000009 |
- |
2-[6-chloro-9-(3-hydroxy-3-methylbut-1-yn-1-yl)-1H-phenanthro[9,10-d]imidazol-2-yl]benzene-1,3-dicarbonitrile |
- |
693551 |
5.3.99.3 | 0.000001 |
- |
(4R)-N-[(1S,3S)-3-(hydroxymethyl)cyclohexyl]-3,3-dimethyl-1-[4-(trifluoromethyl)phenyl]piperidine-4-carboxamide |
pH and temperature not specified in the publication |
747278 |
5.3.99.3 | 0.000001 |
- |
(4S)-N-[(3S)-3-(hydroxymethyl)cyclohexyl]-3,3-dimethyl-1-(8-methylquinolin-2-yl)piperidine-4-carboxamide |
pH and temperature not specified in the publication |
747278 |
5.3.99.3 | 0.000001 |
- |
2-(6-chloro-1H-phenanthro[9,10-d]imidazol-2-yl)benzene-1,3-dicarbonitrile |
- |
693551 |