EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
5.3.99.2 | 0.000021 |
- |
2-phenyl-5-(1H-pyrazol-3-yl)-1,3-thiazole |
37°C |
693542 |
5.3.99.2 | 0.000026 |
- |
N-[5-(1H-indol-4-yl)pyridin-3-yl]-3-(pyridin-3-yl)propanamide |
at 37°C, pH not specified in the publication |
747270 |
5.3.99.2 | 0.000031 |
- |
6-phenoxy-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide |
at 37°C, pH not specified in the publication |
747270 |
5.3.99.2 | 0.000032 |
- |
N-[5-(1H-indol-4-yl)pyridin-3-yl]propanamide |
at 37°C, pH not specified in the publication |
747270 |
5.3.99.2 | 0.000035 |
- |
N-[5-(1H-indol-4-yl)pyridin-3-yl]-5-oxopyrrolidine-2-carboxamide (incorrect configuration definition!) |
at 37°C, pH not specified in the publication |
747270 |
5.3.99.2 | 0.00004 |
- |
3-(3-cyclopropyl-1H-pyrazol-4-yl)-N-ethyl-5,7-dihydro-6H-pyrrolo[3,4-b]pyridine-6-carboxamide |
pH and temperature not specified in the publication |
748543 |
5.3.99.2 | 0.000043 |
- |
N-[5-(1H-indol-4-yl)pyridin-3-yl]-2-(1H-tetrazol-1-yl)acetamide |
at 37°C, pH not specified in the publication |
747270 |
5.3.99.2 | 0.000048 |
- |
6-(piperidin-1-yl)-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide |
at 37°C, pH not specified in the publication |
747270 |
5.3.99.2 | 0.00006 |
- |
6-(3-methoxyphenyl)-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]pyridine-3-carboxamide |
at 37°C, pH not specified in the publication |
747270 |
5.3.99.2 | 0.000071 |
- |
6'-oxo-N-[1-(2,2,2-trifluoroethyl)piperidin-4-yl]-1',6'-dihydro[2,2'-bipyridine]-5-carboxamide |
at 37°C, pH not specified in the publication |
747270 |