EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    4.1.2.27 | 0.000024 |
- |
(R)-1-benzyl-4-(4-(5-cyanopyridin-2-yl)-3-methylpiperazin-1-yl)phthalazine-6-carbonitrile |
at pH 7.4 and 25°C |
748366 |
| 4.1.2.27 | 0.0001 |
- |
(R)-6-(4-(4-benzyl-7-(trifluoromethyl)phthalazin-1-yl)-2-methylpiperazin-1-yl)nicotinonitrile |
at pH 7.4 and 25°C |
748366 |
| 4.1.2.27 | 0.00012 |
- |
N-[2-[(4-butoxy-2,5-dimethylbenzyl)amino]-1-phenylethyl]-5-methyl-1,2-oxazole-3-carboxamide |
pH and temperature not specified in the publication |
747275 |
| 4.1.2.27 | 0.00015 |
- |
N-[1-[4-(3-hydroxyprop-1-yn-1-yl)phenyl]-2-[(4-methoxy-2,5-dimethylbenzyl)amino]ethyl]-5-methyl-1,2-oxazole-3-carboxamide |
pH and temperature not specified in the publication |
747275 |
| 4.1.2.27 | 0.00015 |
- |
N-[1-[4-(4-amino-4-oxobutyl)phenyl]-2-[(4-methoxy-2,5-dimethylbenzyl)amino]ethyl]-5-methyl-1,2-oxazole-3-carboxamide |
pH and temperature not specified in the publication |
747275 |
| 4.1.2.27 | 0.00021 |
- |
(R)-6-(4-(4-benzyl-7-chlorophthalazin-1-yl)-2-methylpiperazin-1-yl)nicotinonitrile |
at pH 7.4 and 25°C |
748366 |
| 4.1.2.27 | 0.00026 |
- |
N-[2-[(4-ethoxy-2,5-dimethylbenzyl)amino]-1-phenylethyl]-5-methyl-1,2-oxazole-3-carboxamide |
pH and temperature not specified in the publication |
747275 |
| 4.1.2.27 | 0.00059 |
- |
N-(2-[[2,5-dimethyl-4-(2,2,2-trifluoroethoxy)benzyl]amino]-1-phenylethyl)-5-methyl-1,2-oxazole-3-carboxamide |
pH and temperature not specified in the publication |
747275 |
| 4.1.2.27 | 0.00072 |
- |
N-[1-(4-fluorophenyl)-2-[(4-methoxy-2,5-dimethylbenzyl)amino]ethyl]-5-methyl-1,2-oxazole-3-carboxamide |
pH and temperature not specified in the publication |
747275 |
| 4.1.2.27 | 0.00073 |
- |
5-cyclopropyl-N-[2-[(4-methoxy-2,5-dimethylbenzyl)amino]-1-phenylethyl]-1,2-oxazole-3-carboxamide |
pH and temperature not specified in the publication |
747275 |
