EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.5.1.52 | 0.0008 |
- |
N,N'-diacetylchitobiosyliodoacetamide |
- |
687514 |
3.5.1.52 | 0.0016 |
- |
Man8GlcNAc2-iodoacetoamide |
- |
687514 |
3.5.1.52 | 0.0017 |
- |
Man9GlcNAc2-iodoacetoamide |
- |
687514 |
3.5.1.52 | 0.0028 |
- |
N,N'-diacetylchitobiosylbromoacetamide |
- |
687514 |
3.5.1.52 | 0.0046 |
- |
carbobenzyloxy-Val-Ala-Asp-alpha-fluoromethylketone |
- |
687444 |
3.5.1.52 | 0.019 |
- |
N,N'-diacetylchitobiosylchloroacetamide |
- |
687514 |
3.5.1.52 | 0.05 |
- |
carbobenzyloxy-Val-Ala-Asp-alpha-fluoromethylketone |
i.e. Z-VAD-fmk, a broad-spectrum caspase inhibitor, IC50: 0.05 mM, binds covalently to the active site of the yeast enzyme, no restoration of enzyme activity by dialysis |
668234 |
3.5.1.52 | 0.17 |
- |
Man9GlcNAc2 |
- |
687514 |