EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.23.5 | 0.0000000783 |
- |
Tb-9 |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.000000126 |
- |
TB-11 |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.000000182 |
- |
tasiamide B |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.00000059 |
- |
pepstatin A |
pH and temperature not specified in the publication |
754469 |
3.4.23.5 | 0.000000693 |
- |
pepstatin A |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.000001 |
- |
pepstatin A |
IC50 of less than 1 nM, at pH 5.5 and 37°C |
731454 |
3.4.23.5 | 0.0000025 |
- |
cathepsin D inhibitor from Streptomyces sp.MBR04 |
in 0.02M sodium citrate, pH 3.0, at 37°C |
731168 |
3.4.23.5 | 0.00000329 |
- |
methyl (5S,8S,11S,12S,16S,19S,22R)-8-(3-amino-3-oxopropyl)-11,22-dibenzyl-12-hydroxy-7,19,21-trimethyl-16-(2-methylpropyl)-3,6,9,14,17,20-hexaoxo-1-phenyl-5-(propan-2-yl)-2-oxa-4,7,10,15,18,21-hexaazatricosan-23-oate |
at pH 3.5 and 25°C |
754470 |
3.4.23.5 | 0.00000584 |
- |
methyl (2S)-1-[(2R,5S,8S,12S,13S)-2,13-dibenzyl-12-hydroxy-15-(3-[(methanesulfonyl)(methyl)amino]-5-[[(1R)-1-phenylethyl]carbamoyl]phenyl)-3,5-dimethyl-8-(2-methylpropyl)-4,7,10,15-tetraoxo-3,6,9,14-tetraazapentadecanan-1-oyl]pyrrolidine-2-carboxylate |
i.e. TB-13, pH and temperature not specified in the publication |
754469 |
3.4.23.5 | 0.00000584 |
- |
TB-13 |
pH and temperature not specified in the publication |
754469 |