EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.51 | 0.000004 |
- |
Nalpha-[(2R,3E)-2-benzyl-4-(phenylsulfonyl)but-3-enoyl]-N-[(4-methylpiperazin-1-yl)carbonyl]-L-phenylalaninamide |
- |
696645 |
3.4.22.51 | 0.000008 |
- |
(2Z)-2-[1-(4-bromophenyl)-2-(3,4-dichlorophenoxy)ethylidene]hydrazine-1-carbothioamide |
23°C, pH 5.5 |
753481 |
3.4.22.51 | 0.000015 |
- |
(2(1H)-pyridinethionato-kappaS2)[2,6-bis[(mercapto-KappaS)methyl]pyridine-kappaN1] oxorhenium(V) |
- |
699388 |
3.4.22.51 | 0.000019 |
- |
(1E)-1-(3,4-dichlorophenyl)pentan-1-one thiosemicarbazone |
IC50: 19 nM |
667951 |
3.4.22.51 | 0.00003 |
- |
(1E)-1-(3,4-dichlorophenyl)propan-1-one thiosemicarbazone |
IC50: 30 nM |
667951 |
3.4.22.51 | 0.00003 |
- |
(1E,2E)-1-(3,4-dichlorophenyl)-3-phenylprop-2-en-1-one thiosemicarbazone |
IC50: 30 nM |
667951 |
3.4.22.51 | 0.00003 |
- |
(1Z)-1-(3,4-dichlorophenyl)-2-phenoxyethan-1-one thiosemicarbazone |
IC50: 30 nM |
667951 |
3.4.22.51 | 0.00003 |
- |
(E)-(3,4-dichlorophenyl)(2-phenylcyclopropyl)methanone thiosemicarbazone |
IC50: 30 nM |
667951 |
3.4.22.51 | 0.00004 |
- |
(1E)-1-(3,4-dichlorophenyl)-3-phenylpropan-1-one thiosemicarbazone |
IC50: 40 nM |
667951 |
3.4.22.51 | 0.00004 |
- |
(E)-(3,4-dichlorophenyl)(4-methylphenyl)methanone thiosemicarbazone |
IC50: 40 nM |
667951 |