EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.39 | 0.0000001 |
- |
N-(2-[[(2-cyanopyrimidin-4-yl)methyl]amino]-2-oxoethyl)-3-[2-(3,5-dichlorophenyl)-2-methylpropanoyl]-4-[(dimethylamino)oxy]benzamide |
isoform AVP5, pH and temperature not specified in the publication |
731464 |
3.4.22.39 | 0.0000001 |
- |
N-(2-[[(2-cyanopyrimidin-4-yl)methyl]amino]-2-oxoethyl)-3-[2-(3,5-dichlorophenyl)-2-methylpropanoyl]-4-[(dimethylamino)oxy]benzamide |
isoform AVP8, pH and temperature not specified in the publication |
731464 |
3.4.22.39 | 0.0000002 |
- |
N-(2-[[(2-cyanopyrimidin-4-yl)methyl]amino]-2-oxoethyl)-3-[2-(3,5-dichlorophenyl)-2-methylpropanoyl]-4-methoxybenzamide |
isoform AVP5, pH and temperature not specified in the publication |
731464 |
3.4.22.39 | 0.0000006 |
- |
N-(2-[[(2-cyanopyrimidin-4-yl)methyl]amino]-2-oxoethyl)-3-[2-(3,5-dichlorophenyl)-2-methylpropanoyl]-4-methoxybenzamide |
isoform AVP8, pH and temperature not specified in the publication |
731464 |
3.4.22.39 | 0.000001 |
- |
3-[2-(3,5-dichlorophenyl)-2-methylpropanoyl]-4-methoxy-N-(2-[[(2E)-3-(methylsulfonyl)prop-2-en-1-yl]amino]-2-oxoethyl)benzamide |
isoform AVP5, pH and temperature not specified in the publication |
731464 |
3.4.22.39 | 0.000001 |
- |
3-[2-(3,5-dichlorophenyl)-2-methylpropanoyl]-4-methoxy-N-(2-[[(2E)-3-(methylsulfonyl)prop-2-en-1-yl]amino]-2-oxoethyl)benzamide |
isoform AVP8, pH and temperature not specified in the publication |
731464 |
3.4.22.39 | 0.000001 |
- |
N-[(2S)-2-(3,5-dichlorophenyl)-2-(ethylamino)acetyl]-3-methyl-L-valylglycyl-N-[(2E)-3-(methylsulfonyl)prop-2-en-1-yl]glycinamide |
IC50 below 0.000001 mM, isoform AVP8, pH and temperature not specified in the publication |
731464 |
3.4.22.39 | 0.000002 |
- |
(2S)-2-(3,5-dichlorophenyl)-N-[(3S)-1-[2-[(2-[[(2E)-3-(methylsulfonyl)prop-2-en-1-yl]amino]-2-oxoethyl)amino]-2-oxoethyl]-2-oxopyrrolidin-3-yl]butanamide |
isoform AVP5, pH and temperature not specified in the publication |
731464 |
3.4.22.39 | 0.000004 |
- |
(2S)-2-(3,5-dichlorophenyl)-N-[(3S)-1-[2-[(2-[[(2E)-3-(methylsulfonyl)prop-2-en-1-yl]amino]-2-oxoethyl)amino]-2-oxoethyl]-2-oxopyrrolidin-3-yl]butanamide |
isoform AVP8, pH and temperature not specified in the publication |
731464 |
3.4.22.39 | 0.000007 |
- |
N-[2-[(cyanomethyl)amino]-2-oxoethyl]-3-[2-(3,5-dichlorophenyl)-2-methylpropanoyl]-4-[(dimethylamino)oxy]benzamide |
isoform AVP5, pH and temperature not specified in the publication |
731464 |