EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.4.21.91 | 0.000019 |
- |
2,6-difluoro-benzoyl-Nle-Lys-Arg-Arg-CF3-ketone |
pH 7.4, temperature not specified in the publication, versus the linked NS2B-NS3 complex |
755305 |
| 3.4.21.91 | 0.000038 |
- |
benzoyl-Nle-Lys-Arg-Arg-B(OH)2 |
pH 7.4, temperature not specified in the publication, versus the linked NS2B-NS3 complex |
755305 |
| 3.4.21.91 | 0.000056 |
- |
4-phenylphenylacetyl-Lys-Lys-Arg |
pH 8.5, 20°C |
717102 |
| 3.4.21.91 | 0.0001024 |
- |
Aprotinin |
- |
677891 |
| 3.4.21.91 | 0.000105 |
- |
SID-852843 |
in 10 mM Tris-HCl buffer, pH 8.0, containing 20% (v/v) glycerol and 0.005% Brij 35 |
707680 |
| 3.4.21.91 | 0.000105 |
- |
[5-amino-1-(4-methoxyphenyl)sulfonylpyrazol-3-yl] benzoate |
- |
677891 |
| 3.4.21.91 | 0.00011 |
- |
SID-4245669 |
in 10 mM Tris-HCl buffer, pH 8.0, containing 20% (v/v) glycerol and 0.005% Brij 35 |
707680 |
| 3.4.21.91 | 0.00011 |
- |
[5-amino-1-(4-methoxyphenyl)sulfonylpyrazol-3-yl] thiophene-2-carboxylate |
- |
677891 |
| 3.4.21.91 | 0.000208 |
- |
(S)-2-acetamido-6-amino-N-((S)-5-guanidino-1-oxopentan-2-yl)hexanamide |
pH and temperature not specified in the publication |
755564 |
| 3.4.21.91 | 0.000297 |
- |
[5-amino-1-(4-methoxyphenyl)sulfonylpyrazol-3-yl] 2-bromobenzoate |
- |
677891 |
