EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.21.77 | 0.000001 |
- |
AUY922 |
- |
708155 |
3.4.21.77 | 0.00025 |
- |
R/S-diphenyl[N-benzyloxycarbonylamino(4-carbamoylphenyl)methyl]phosphonate |
pH and temperature not specified in the publication |
732227 |
3.4.21.77 | 0.0003 |
- |
2-(2-methyl-3-nitrophenyl)-4H-3,1-benzoxazin-4-one |
- |
701037 |
3.4.21.77 | 0.00034 |
- |
benzyl 1-(2-(3-(benzyloxycarbonyl)phenyl)acetyl)-3-(4-hydroxybenzyl)-4-oxoazetidine-2-carboxylate |
- |
682769 |
3.4.21.77 | 0.0005 |
- |
(5-amino-3-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl)(3,4-dimethoxyphenyl)methanone |
- |
701037 |
3.4.21.77 | 0.0009 |
- |
(5-amino-3-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl)(4-methoxyphenyl)methanone |
- |
701037 |
3.4.21.77 | 0.0011 |
- |
(2S,3S)-ethyl 3-benzyl-4-oxo-1-tosylazetidine-2-carboxylate |
- |
682769 |
3.4.21.77 | 0.00143 |
- |
benzyl 3-benzyl-1-(2-(3-(benzyloxycarbonyl)phenyl)acetyl)-4-oxoazetidine-2-carboxylate |
- |
682769 |
3.4.21.77 | 0.0022 |
- |
(3-benzyl-1-(ethylsulfonyl)-4-oxoazetidin-2-yl)methyl benzoate |
- |
682769 |
3.4.21.77 | 0.0022 |
- |
(5-amino-3-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl)(4-chlorophenyl)methanone |
- |
701037 |