EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.4.21.68 | -999 |
- |
xenon |
although xenon at 25% (v/v) has no effect, xenon at higher concentrations of 37.5, 50 and 75% inhibit the catalytic efficiencies of human enzyme, IC50 is 34.85% (v/v) |
709252 |
| 3.4.21.68 | -999 |
- |
xenon |
although xenon at 25% (v/v) has no effect, xenon at higher concentrations of 37.5, 50 and 75% inhibit the catalytic efficiencies of murine enzyme, IC50 is 37.39% (v/v) |
709252 |
| 3.4.21.68 | 0.0000223 |
- |
Chi-tPA 2 |
pH 7.4-8.5, 37°C, recombinant chimeric enzyme |
755312 |
| 3.4.21.68 | 0.0000289 |
- |
Chi-tPA 1 |
pH 7.4-8.5, 37°C, recombinant chimeric enzyme |
755312 |
| 3.4.21.68 | 0.000197 |
- |
Chi-tPA 3 |
pH 7.4-8.5, 37°C, recombinant chimeric enzyme |
755312 |
| 3.4.21.68 | 0.0002 |
- |
Chi-tPA 4 |
pH 7.4-8.5, 37°C, recombinant chimeric enzyme |
755312 |
| 3.4.21.68 | 0.00021 |
- |
Chi-tPA 5 |
pH 7.4-8.5, 37°C, recombinant chimeric enzyme |
755312 |
| 3.4.21.68 | 0.0034 |
- |
N2-(3'-(trifluoromethyl)biphenyl-4-yl)naphthalene-2,6-dicarboxamide |
pH 7.4-8.3, 37°C |
731467 |
| 3.4.21.68 | 0.0036 |
- |
4-(2-aminoethoxy)-N-[3-chloro-2-ethoxy-5-(piperidin-1-yl)phenyl]-3,5-dimethylbenzamide |
pH 7.4-8.3, 37°C |
731467 |
| 3.4.21.68 | 0.0039 |
- |
2-([6-[(3'-carbamimidoylbiphenyl-3-yl)oxy]-3,5-difluoro-4-methylpyridin-2-yl]oxy)-4-(dimethylamino)benzoic acid |
pH 7.4-8.3, 37°C |
731467 |
