EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.4.21.21 | 0.000000022 |
- |
VLCWTWETCER-NH2 |
IC50: 0.022 nM |
654613 |
| 3.4.21.21 | 0.00000023 |
- |
EEWEVLCWTWETCERGEGVEEELWEWR |
maximal inhibition to 99%, IC50: 230 pM |
656136 |
| 3.4.21.21 | 0.0000015 |
- |
EEWEVLCWTWETCER |
maximal inhibition to 74%, IC50: 1.5 nM |
656136 |
| 3.4.21.21 | 0.0000015 |
- |
EEWEVLCWTWETCERGEG-NH2 |
IC50: 1.5 nM |
654613 |
| 3.4.21.21 | 0.0000016 |
- |
EEWEVLCWTWETCER |
IC50: 1.6 nM, partial hyperbolic mixed-type inhibitor of factor X activation, partial competitive inhibitor of amidolytic activity. Inhibits activation of factor X and factor IX and amidolytic activity of Chromozym t-PA with IC50 values of 1.6 nM, 3.5 nM |
654613 |
| 3.4.21.21 | 0.0000025 |
- |
WEVLCWTWETCER-NH2 |
IC50: 2.5 nM |
654613 |
| 3.4.21.21 | 0.0000038 |
- |
EEWEVLCWTWETCERGEG-(Z-domain of protein A) |
IC50: 3.8 nM |
654613 |
| 3.4.21.21 | 0.0000048 |
- |
EWEVLCWTWETCERGE-(Z-domain of protein A) |
IC50: 4.8 nM |
654613 |
| 3.4.21.21 | 0.0000059 |
- |
MEEWEVLCWTWETCERGEGQ-(Z-domain of protein A) |
IC50: 5.9 nM |
654613 |
| 3.4.21.21 | 0.000016 |
- |
3-amino-5-[1-[2-([4-[amino(imino)methyl]benzyl]amino)-2-oxoethyl]-3-chloro-5-(isopropylamino)-6-oxo-1,6-dihydropyrazin-2-yl]benzoic acid |
pH 8.0, IC50: 16 nM, potent and highly selective inhibitor, selectivity versus factor Xa and thrombin |
656463 |
