EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.21.113 | 0.00013 |
- |
12-cyclohexyl-5,5-dimethyl-11,14-dioxo-2,6-dioxa-10,13-diazatricyclo[14.3.1.17,10]henicosa-1(19),16(20),17-triene-9-carboxylic acid ((([1-(dimethylcarbamoylphenylmethyl)carbamoyl]-methyl)aminooxalyl)butyl)amide |
- |
669812 |
3.4.21.113 | 0.00024 |
- |
12-cyclohexyl-11,14-dioxo-2,6-dioxa-10,13-diazatricyclo[14.3.1.17,10]henicosa-1(19),16(20),17-triene-9-carboxylic acid ((([1-(dimethylcarbamoylphenylmethyl)carbamoyl]methyl)aminooxalyl)butyl)amide |
S-isomer |
669812 |
3.4.21.113 | 0.00068 |
- |
1-O-(3-O-galloylgalloyl)-2,3,4-tri-O-galloyl-beta-D-glucose |
- |
685513 |
3.4.21.113 | 0.00077 |
- |
3,3'-digalloylproprodelphinidin B2 |
- |
684506 |
3.4.21.113 | 0.0008 |
- |
2-O-(4-O-galloylgalloyl)-1,3,4-tri-O-galloyl-beta-D-glucose |
- |
685513 |
3.4.21.113 | 0.00091 |
- |
3,3'-digalloylprocyanidin B2 |
- |
684506 |
3.4.21.113 | 0.001 |
- |
1,3,4-tri-O-galloyl-beta-D-glucose |
- |
685513 |
3.4.21.113 | 0.0047 |
- |
4-phenylphenacetyl-L-Lys-L-Lys-agmatine |
at pH 8.0 in Tris-HCl (10 mM), CHAPS (1 mM) and glycerol (20% v/v), at 25°C |
717569 |
3.4.21.113 | 0.00851 |
- |
epigallocatechin-3-O-gallate |
- |
684506 |
3.4.21.113 | 0.01009 |
- |
1,3,6-tri-O-galloyl-beta-D-glucose |
- |
685513 |