EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.2.1.113 | 0.00005 |
0.0001 |
kifunensine |
at pH 7.0 and 30°C |
753758 |
3.2.1.113 | 0.00035 |
- |
kifunensine |
37°C, pH 6.0, substrate methyl 2-O-alpha-D-mannopyranosyl-alpha-D-mannopyranoside |
751841 |
3.2.1.113 | 0.00047 |
- |
kifunensine |
37°C, pH 6.0, substrate methyl 2-O-alpha-D-mannopyranosyl-alpha-D-mannopyranoside |
751841 |
3.2.1.113 | 0.003 |
- |
D-mannonolactam amidrazone |
pH not specified in the publication, temperature not specified in the publication |
754043 |
3.2.1.113 | 0.004 |
- |
D-mannonolactam amidrazone |
pH not specified in the publication, temperature not specified in the publication |
754043 |
3.2.1.113 | 0.03 |
- |
1-deoxymannojirimycin |
37°C, pH 6.0, substrate methyl 2-O-alpha-D-mannopyranosyl-alpha-D-mannopyranoside |
751841 |
3.2.1.113 | 0.04 |
- |
1-deoxymannojirimycin |
37°C, pH 6.0, substrate methyl 2-O-alpha-D-mannopyranosyl-alpha-D-mannopyranoside |
751841 |
3.2.1.113 | 0.19 |
- |
1-deoxymannojirimycin |
at pH 6.0 and 37°C |
754617 |
3.2.1.113 | 0.23 |
- |
1-deoxymannojirimycin |
at pH 6.0 in 50 mM Tris-MES and at 37°C |
753587 |
3.2.1.113 | 0.47 |
- |
swainsonine |
at pH 6.0 in 50 mM Tris-MES and at 37°C |
753587 |