EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.1.4.39 | 0.000013 |
- |
[3-([4-[(5Z)-5-(3,4-dichlorobenzylidene)-4-oxo-4,5-dihydro-1,3-thiazol-2-yl]piperazin-1-yl]methyl)phenyl]boronic acid |
pH 9.0, 37°C |
728853 |
| 3.1.4.39 | 0.000016 |
- |
lysophosphatidic acid |
reported as an inhibitor of its own production, incubating human autotaxin gamma with lysophosphatidic acid |
680925 |
| 3.1.4.39 | 0.000017 |
- |
lysophosphatidic acid |
reported as an inhibitor of its own production, incubating human autotaxin beta with lysophosphatidic acid |
680925 |
| 3.1.4.39 | 0.000018 |
- |
lysophosphatidic acid |
reported as an inhibitor of its own production, incubating murine autotaxin beta with lysophosphatidic acid |
680925 |
| 3.1.4.39 | 0.00002 |
- |
lysophosphatidic acid |
reported as an inhibitor of its own production, incubating murine autotaxin gamma with lysophosphatidic acid |
680925 |
| 3.1.4.39 | 0.000022 |
- |
[4-([4-[(5Z)-5-(3,4-dichlorobenzylidene)-4-oxo-4,5-dihydro-1,3-thiazol-2-yl]piperazin-1-yl]methyl)phenyl]boronic acid |
pH 9.0, 37°C |
728853 |
| 3.1.4.39 | 0.000025 |
- |
(5Z)-5-(3,4-dichlorobenzylidene)-2-[4-[4-(dihydroxymethyl)benzyl]piperazin-1-yl]-1,3-thiazol-4(5H)-one |
pH 9.0, 37°C |
728853 |
| 3.1.4.39 | 0.000028 |
- |
[3-[(4-[(Z)-[3-(4-fluorobenzyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]phenoxy)methyl]phenyl]boronic acid |
in Tris-HCl buffer (pH 7.4) at 37°C |
706564 |
| 3.1.4.39 | 0.000038 |
- |
lysophosphatidic acid |
reported as an inhibitor of its own production, incubating human autotaxin alpha with lysophosphatidic acid |
680925 |
| 3.1.4.39 | 0.000038 |
- |
lysophosphatidic acid |
reported as an inhibitor of its own production, incubating murine autotaxin alpha with lysophosphatidic acid |
680925 |
