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EC Number	IC50 Value	IC50 Value Maximum	Inhibitor	Commentary	Reference
2.8.2.2	0.00006	-	bazedoxifene N-oxide	liver cytosol, pH 7.4, 37°C, substrate lithocholic acid	761727
2.8.2.2	0.00008	-	arzoxifene	liver cytosol, pH 7.4, 37°C, substrate taurolithocholic acid	761727
2.8.2.2	0.00013	-	bazedoxifene	liver cytosol, pH 7.4, 37°C, substrate taurolithocholic acid	761727
2.8.2.2	0.00015	-	Pentachlorophenol	in 0.1 M sodium phosphate, pH 7.2, and 2 mM EDTA for 30 min at 16°C	703834
2.8.2.2	0.00016	-	des(1-azepanyl)ethylbazedoxifene	liver cytosol, pH 7.4, 37°C, substrate lithocholic acid	761727
2.8.2.2	0.00016	-	pentabromophenol	in 0.1 M sodium phosphate, pH 7.2, and 2 mM EDTA for 30 min at 16°C	703834
2.8.2.2	0.00018	-	raloxifene	liver cytosol, pH 7.4, 37°C, substrate taurolithocholic acid	761727
2.8.2.2	0.0002	-	arzoxifene	liver cytosol, pH 7.4, 37°C, substrate glycolithocholic acid	761727
2.8.2.2	0.00021	-	bazedoxifene	liver cytosol, pH 7.4, 37°C, substrate lithocholic acid	761727
2.8.2.2	0.00021	-	triiodophenol	in 0.1 M sodium phosphate, pH 7.2, and 2 mM EDTA for 30 min at 16°C	703834

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Release 2023.1 (January 2023)