EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.7.86 | 0.00023 |
- |
6-(4-(2-aminophenyl)-1H-1,2,3-triazol-1-yl)-N2-(4-iodophenyl)-1,3,5-triazine-2,4-diamine |
pH 7.5, 37°C |
761723 |
2.7.7.86 | 0.00024 |
0.00027 |
methyl 4-amino-6-((3,4,5-trifluorophenyl)amino)-1,3,5-triazine-2-carboxylate |
pH 7.5, 37°C |
761723 |
2.7.7.86 | 0.00045 |
0.00066 |
methyl 4-amino-6-((4-iodophenyl)amino)-1,3,5-triazine-2-carboxylate |
pH 7.5, 37°C |
761723 |
2.7.7.86 | 0.00059 |
- |
4-amino-6-((4-iodophenyl)amino)-1,3,5-triazine-2-carboxylicacid |
pH 7.5, 37°C |
761723 |
2.7.7.86 | 0.0014 |
- |
methyl 4-amino-6-((4-ethynylphenyl)amino)-1,3,5-triazine-2-carboxylate |
pH 7.5, 37°C |
761723 |
2.7.7.86 | 0.0015 |
- |
methyl 4-amino-6-[(3,5-difluoro-4-iodophenyl)amino]-1,3,5-triazine-2-carboxylate |
pH 7.5, 37°C |
761723 |
2.7.7.86 | 0.0023 |
- |
6-(aminomethyl)-N2-(4-fluorophenyl)-1,3,5-triazine-2,4-diamine |
pH 7.5, 37°C |
761723 |
2.7.7.86 | 0.0025 |
- |
N-2-(4-iodophenyl)-6-(1,3,4-oxadiazol-2-yl)-1,3,5-triazine-2,4-diamine |
pH 7.5, 37°C |
761723 |
2.7.7.86 | 0.0034 |
- |
N2-(4-iodophenyl)-6-(1H-pyrazol-1-yl)-1,3,5-triazine-2,4-diamine |
pH 7.5, 37°C |
761723 |
2.7.7.86 | 0.0038 |
- |
4-amino-6-(4-fluoroanilino)-1,3,5-triazine-2-carboxylic acid |
pH 7.5, 37°C |
761723 |