EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.6.1 | 0.05 |
- |
Ca2+ |
IC50 of 0.05 mM |
642711 |
2.7.6.1 | 0.07 |
- |
ADP |
in 50 mM Tris-HCl pH 8.0, at 25°C |
723571 |
2.7.6.1 | 0.07 |
- |
ADP |
mutant enzyme D58H, in 50 mM potassium phosphate at pH 7.5, 5 mM MgCl2, at 37°C |
721377 |
2.7.6.1 | 0.08 |
- |
ADP |
wild type enzyme, in 50 mM potassium phosphate at pH 7.5, 5 mM MgCl2, at 37°C |
721377 |
2.7.6.1 | 0.174 |
- |
ADP |
pH 7.5, 25°C |
762221 |
2.7.6.1 | 0.4 |
- |
GDP |
in 50 mM potassium phosphate pH 8.0, at 37°C |
723524 |
2.7.6.1 | 0.44 |
- |
ADP |
mutant enzyme N120S, in 50 mM potassium phosphate at pH 7.5, 5 mM MgCl2, at 37°C |
721377 |
2.7.6.1 | 0.45 |
- |
GDP |
wild type enzyme, in 50 mM potassium phosphate at pH 7.5, 5 mM MgCl2, at 37°C |
721377 |
2.7.6.1 | 0.51 |
- |
GDP |
mutant enzyme D58H, in 50 mM potassium phosphate at pH 7.5, 5 mM MgCl2, at 37°C |
721377 |
2.7.6.1 | 0.84 |
- |
ADP |
mutant enzyme L135I, in 50 mM potassium phosphate at pH 7.5, 5 mM MgCl2, at 37°C |
721377 |