EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.11.24 | -999 |
- |
(2S)-2-([6-[(2-aminobenzyl)amino]-9-(1-methylethyl)-9H-purin-2-yl]amino)butan-1-ol |
relative activity, 58% of control |
702773 |
2.7.11.24 | -999 |
- |
2,2'-[[6-(benzylamino)-9-(1-methylethyl)-9H-purin-2-yl]imino]diethanol |
relative activity, 37% of control |
702773 |
2.7.11.24 | -999 |
- |
2-(2-[[6-(benzylamino)-9-(1-methylethyl)-9H-purin-2-yl]amino]ethoxy)ethanol |
relative activity, 56% of control |
702773 |
2.7.11.24 | -999 |
- |
2-(4-fluorophenyl)-3-(pyridin-4-yl)pyrido[2,3-b]pyrazine |
46% at 10 microM |
705058 |
2.7.11.24 | -999 |
- |
2-(4-fluorophenyl)-3-pyridin-4-ylpyrido[3,4-b]pyrazine |
33% at 10 microM, mixture of 3-(4-fluorophenyl)-2-pyridin-4-ylpyrido[3,4-b]pyrazine and 2-(4-fluorophenyl)-3-pyridin-4-ylpyrido[3,4-b]pyrazine |
705058 |
2.7.11.24 | -999 |
- |
2-(4-fluorophenyl)-6-methoxy-3-(pyridin-4-yl)quinoxaline |
33% at 10 microM |
705058 |
2.7.11.24 | -999 |
- |
2-([6-[(3-methylbut-2-en-1-yl)amino]-9-(1-methylethyl)-9H-purin-2-yl]amino)ethanol |
relative activity, 96% of control |
702773 |
2.7.11.24 | -999 |
- |
2-([9-methyl-6-[(3-methylbut-2-en-1-yl)amino]-9H-purin-2-yl]amino)ethanol |
relative activity, 44% of control |
702773 |
2.7.11.24 | -999 |
- |
2-([[2-[[(1S)-1-(hydroxymethyl)propyl]amino]-9-(1-methylethyl)-9H-purin-6-yl]amino]methyl)phenol |
relative activity, 23% of control |
702773 |
2.7.11.24 | -999 |
- |
2-([[2-[[1-(hydroxymethyl)-2-methylbutyl]amino]-9-(1-methylethyl)-9H-purin-6-yl]amino]methyl)phenol |
relative activity, 50% of control |
702773 |