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EC Number
IC50 Value
IC50 Value Maximum
Inhibitor
Commentary
Reference
2.7.11.16
0.00004
0.00005
Ca2+/calmodulin
inhibit GRK5 with an IC50 of 40-50 nM, inhibition mechanism via inducing inhibitory autophosphorylation and blocking of membrane association
662911
2.7.11.16
0.000079
-
RNA aptamer C13
inhibition of GRK5
690032
2.7.11.16
0.00008
-
Calmodulin
reaction of isoenzyme GRK4alpha with rhodopsin, IC50: 80 nM
491135
2.7.11.16
0.0011
-
CCG-265328
at pH 7.5, and temperature not specified in the publication
760266
2.7.11.16
0.0025
-
GSK1326255A
at pH 7.5, and temperature not specified in the publication
760266
2.7.11.16
0.0032
-
GSK1713088A
at pH 7.5, and temperature not specified in the publication
760266
2.7.11.16
0.0032
-
GSK2163632A
at pH 7.5, and temperature not specified in the publication
760266
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