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EC Number IC50 Value IC50 Value Maximum Inhibitor Commentary Reference
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.120.00000013 - N-(cyclopropylmethyl)-4-[7-[(dimethylamino)methyl]-2-[3-(methanesulfonyl)phenyl]imidazo[1,2-a]pyridin-3-yl]pyrimidin-2-amine wild type enzyme, at pH 7.4 and 25°C 761994
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.120.00000016 - N-[5-(3-[2-[(cyclopropylmethyl)amino]pyrimidin-4-yl]-7-[(dimethylamino)methyl]-6-methylimidazo[1,2-a]pyridin-2-yl)-2-fluorophenyl]methanesulfonamide wild type enzyme, at pH 7.4 and 25°C 761994
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.120.00000045 - 4-[7-[(dimethylamino)methyl]-2-(4-fluorophenyl)-6-methylimidazo[1,2-a]pyridin-3-yl]-N-[4-(piperazin-1-yl)phenyl]pyrimidin-2-amine wild type enzyme, at pH 7.4 and 25°C 761994
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.120.00000079 - 4-[7-[(dimethylamino)methyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]-N-[4-(piperazin-1-yl)phenyl]pyrimidin-2-amine wild type enzyme, at pH 7.4 and 25°C 761994
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.120.00000079 - N-(5-[3-(2-aminopyrimidin-4-yl)-7-[(dimethylamino)methyl]imidazo[1,2-a]pyridin-2-yl]-2-fluorophenyl)methanesulfonamide wild type enzyme, at pH 7.4 and 25°C 761994
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.120.00000088 - 4-[7-[(dimethylamino)methyl]-2-[3-(methanesulfonyl)phenyl]imidazo[1,2-a]pyridin-3-yl]pyrimidin-2-amine wild type enzyme, at pH 7.4 and 25°C 761994
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.120.000001 - 4-[2-(4-fluorophenyl)-5-(1-methylpiperidin-4-yl)-1H-pyrrol-3-yl]pyridine - 675507
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.120.000001 - 4-[2-(fluorophenyl)-5-(1-methylpiperidine-4-yl)-1H-pyrrol-3-yl]pyridine inhibitor of apicomplexan parasite enzyme, IC50 is 1 nM for the enzyme of Eimeria tenella, mechanism 661813
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.120.00000119 - N-(5-[3-(2-aminopyrimidin-4-yl)-7-[(dimethylamino)methyl]-6-methylimidazo[1,2-a]pyridin-2-yl]-2-fluorophenyl)methanesulfonamide wild type enzyme, at pH 7.4 and 25°C 761994
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.120.00000155 - 4-[2-(fluorophenyl)-5-(1-methylpiperidine-4-yl)-1H pyrrol-3-yl] pyridine mutant enzyme T618M, in 50 mM HEPES, at pH 7.4, at 30°C 694797
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