EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    2.6.1.7 | 0.000004 |
- |
(3S)-3-amino-6-benzyl-1-hydroxy-7-methoxy-3,4-dihydroquinolin-2(1H)-one |
mass spectrometry assay, pH 7.5, temperature not specified in the publication |
737437 |
| 2.6.1.7 | 0.000005 |
- |
(3S)-3-amino-6-benzyl-1-hydroxy-7-methoxy-3,4-dihydroquinolin-2(1H)-one |
fluorescence assay, pH 7.5, temperature not specified in the publication |
737437 |
| 2.6.1.7 | 0.000015 |
- |
(3S)-3-amino-1-hydroxy-3,4-dihydroquinolin-2(1H)-one |
flourescence assay, pH 7.5, temperature not specified in the publication |
737437 |
| 2.6.1.7 | 0.00003 |
- |
(3S)-3-amino-1-hydroxy-3,4-dihydroquinolin-2(1H)-one |
mass spectrometry assay, pH 7.5, temperature not specified in the publication |
737437 |
| 2.6.1.7 | 0.00081 |
- |
N-(3-chloro-4-methylphenyl)-8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide |
pH and temperature not specified in the publication |
758920 |
| 2.6.1.7 | 0.00091 |
- |
(S)-(-)-9-(4-aminopiperazin-1-yl)-8-fluoro-3-methyl-6-oxo-2,3-dihydro-6H-1-oxa-3a-azaphenalene-5-carboxylic acid |
0.0015 mM or the two enantiomers, pH 8.0, 37°C |
722912 |
| 2.6.1.7 | 0.002 |
- |
cysteine sulfinate |
pH 7.5, 25°C |
722236 |
| 2.6.1.7 | 0.0024 |
- |
(6R)-N-(3-chloro-4-fluorophenyl)-8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide |
pH and temperature not specified in the publication |
758920 |
| 2.6.1.7 | 0.0039 |
- |
carbenoxolone |
isoform KAT2, at pH 9.5 and 37°C |
760173 |
| 2.6.1.7 | 0.0045 |
- |
(6R)-8-cyclopropyl-N-(3,5-dimethylphenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide |
pH and temperature not specified in the publication |
758920 |
