EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.4.2.2 | 0.000003 |
- |
5-benzylacyclouridine |
substrate uridine, pH 7.6, 37°C |
721540 |
2.4.2.2 | 0.000005 |
- |
5-benzylacyclouridine |
substrate deoxythymidine, pH 7.6, 37°C |
721540 |
2.4.2.2 | 0.03 |
- |
7-deazaxanthine |
substrate deoxythymidine, pH 7.6, 37°C |
721540 |
2.4.2.2 | 0.06 |
- |
7-deazaxanthine |
substrate uridine, pH 7.6, 37°C |
721540 |
2.4.2.2 | 0.113 |
- |
3,5-bis-(4-chlorobenzoyl)-alpha-D-ribose 1-phosphate |
substrate deoxythymidine, pH 7.6, 37°C |
721554 |
2.4.2.2 | 0.128 |
- |
3,5-bis-(4-chlorobenzoyl)-alpha-D-ribose 1-phosphate |
substrate 5-fluorodeoxyuridine, pH 7.6, 37°C |
721554 |
2.4.2.2 | 0.159 |
- |
3,5-bis-(4-chlorobenzoyl)-alpha-D-ribose 1-phosphate |
substrate 5-iododeoxyuridine pH 7.6, 37°C |
721554 |
2.4.2.2 | 0.188 |
- |
3,5-bis-(4-chlorobenzoyl)-alpha-D-ribose 1-phosphate |
substrate uridine, pH 7.6, 37°C |
721554 |
2.4.2.2 | 0.5 |
- |
5-chloro-6-(1-[2-iminopyrrolidinyl]methyl)uracil |
substrate deoxythymidine, pH 7.6, 37°C |
721540 |
2.4.2.2 | 0.5 |
- |
5-chloro-6-(1-[2-iminopyrrolidinyl]methyl)uracil |
substrate uridine, pH 7.6, 37°C |
721540 |