EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   2.4.1.227 | 0.00096 |
- |
ristocetin A |
pH 8.0, 37°C |
758570 |
| 2.4.1.227 | 0.0014 |
- |
(5E)-5-[(4-tert-butylphenyl)methylidene]-3-[(4-methylpiperidin-1-yl)methyl]-2-sulfanylidene-1,3-thiazolidin-4-one |
pH 7.9, temperature not specified in the publication |
758938 |
| 2.4.1.227 | 0.0014 |
- |
5-(3-[(E)-[1-(3-chlorophenyl)-2,4,6-trioxo-1,3-diazinan-5-ylidene]methyl]-2,5-dimethyl-1H-pyrrol-1-yl)benzene-1,3-dicarboxylic acid |
pH 7.9, temperature not specified in the publication |
758938 |
| 2.4.1.227 | 0.0014 |
- |
ristocetin A |
pH 8.0, 37°C |
758570 |
| 2.4.1.227 | 0.002 |
- |
ToXa-1 |
pH 8.0, 37°C |
758570 |
| 2.4.1.227 | 0.0034 |
- |
[(5E)-5-[(3-bromo-5-chloro-2-hydroxyphenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetic acid |
pH 7.9, temperature not specified in the publication |
758938 |
| 2.4.1.227 | 0.0035 |
- |
2-[(5Z)-5-(1-benzyl-5-bromo-2-oxo-1,2-dihydro-3H-indol-3-ylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]ethane-1-sulfonic acid |
pH 7.9, temperature not specified in the publication |
758938 |
| 2.4.1.227 | 0.0035 |
- |
PyDT-1 |
pH 8.0, 37°C |
758570 |
| 2.4.1.227 | 0.004 |
- |
5-([3-[2-(4-tert-butylphenoxy)ethoxy]phenyl]methylidene)-2-sulfanylidene-1,3-diazinane-4,6-dione |
pH 7.9, temperature not specified in the publication |
758938 |
| 2.4.1.227 | 0.0054 |
- |
3-[[(3E)-3-[[5-(4-bromophenyl)furan-2-yl]methylidene]-2-oxo-5-phenyl-2,3-dihydro-1H-pyrrol-1-yl]methyl]benzoic acid |
pH 7.9, temperature not specified in the publication |
758938 |
