EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    2.4.1.17 | -999 |
- |
more |
inhibition of isozyme UGT2B7 at several different concentration of inhibitor compounds |
691812 |
| 2.4.1.17 | 0.000045 |
- |
regorafenib |
isoform UGT1A1, at pH 7.4, temperature not specified in the publication |
756020 |
| 2.4.1.17 | 0.000066 |
- |
sorafenib |
isoform UGT1A1, at pH 7.4, temperature not specified in the publication |
756020 |
| 2.4.1.17 | 0.00007 |
- |
(R)-cyclopropyl(phenyl)methanol |
IC50: 0.00007 mM |
675319 |
| 2.4.1.17 | 0.0001 |
- |
isolongifolol |
IC50: 0.0001 mM |
675319 |
| 2.4.1.17 | 0.00013 |
- |
2,4-Dibromophenol |
isoform UGT1A7, at pH 7.4 and 37°C |
756487 |
| 2.4.1.17 | 0.00014 |
- |
2,5-dibromophenol |
isoform UGT2B7, at pH 7.4 and 37°C |
756487 |
| 2.4.1.17 | 0.00015 |
- |
2,5-dibromophenol |
isoform UGT1A9, at pH 7.4 and 37°C |
756487 |
| 2.4.1.17 | 0.00018 |
- |
3,5-dibromophenol |
isoform UGT1A9, at pH 7.4 and 37°C |
756487 |
| 2.4.1.17 | 0.000187 |
- |
pazopanib |
isoform UGT1A8, at pH 7.4, temperature not specified in the publication |
756020 |
