EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.3.1.61 | 0.00351 |
- |
2-(4-fluorophenyl)-5-(methanesulfonyl)-1,3,4-oxadiazole |
at pH 7.2 and 28° |
757052 |
2.3.1.61 | 0.00358 |
- |
2-(4-fluoro-3-[[(prop-2-yn-1-yl)oxy]methyl]phenyl)-5-(methanesulfonyl)-1,3,4-oxadiazole |
at pH 7.2 and 28° |
757052 |
2.3.1.61 | 0.00358 |
- |
2-(methylsulfonyl)-5-(4-fluoro-3-((prop-2-yn-1-yloxy)methyl)-phenyl)-1,3,4-oxadiazole |
at pH 7.2 and 28°C |
757052 |
2.3.1.61 | 0.00399 |
- |
2-(2,4-dichloro-3-[[(prop-2-yn-1-yl)oxy]methyl]phenyl)-5-(methanesulfonyl)-1,3,4-oxadiazole |
at pH 7.2 and 28° |
757052 |
2.3.1.61 | 0.00551 |
- |
2-(methanesulfonyl)-5-(4-[[(prop-2-yn-1-yl)oxy]methyl]phenyl)-1,3,4-oxadiazole |
at pH 7.2 and 28° |
757052 |
2.3.1.61 | 0.0068 |
- |
2-(2,4-dichloro-3-[[(prop-2-yn-1-yl)oxy]methyl]phenyl)-5-(ethanesulfonyl)-1,3,4-oxadiazole |
at pH 7.2 and 28° |
757052 |
2.3.1.61 | 0.00706 |
- |
2-(ethanesulfonyl)-5-(4-fluoro-3-[[(prop-2-yn-1-yl)oxy]methyl]phenyl)-1,3,4-oxadiazole |
at pH 7.2 and 28° |
757052 |
2.3.1.61 | 0.00795 |
- |
2-(ethanesulfonyl)-5-(4-fluoro-3-[[(prop-2-yn-1-yl)oxy]methyl]phenyl)-1,3,4-oxadiazole |
at pH 7.2 and 28° |
757052 |
2.3.1.61 | 0.00859 |
- |
2-(4-fluorophenyl)-5-(methanesulfonyl)-1,3,4-oxadiazole |
at pH 7.2 and 28° |
757052 |
2.3.1.61 | 0.01263 |
- |
2-(ethanesulfonyl)-5-(4-[[(prop-2-yn-1-yl)oxy]methyl]phenyl)-1,3,4-oxadiazole |
at pH 7.2 and 28° |
757052 |