EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.1.2.3 | -999 |
- |
N-(4-[[(2,4-diaminopteridin-6-yl)methyl](methyl)amino]benzoyl)glutamic acid |
value above 0.05 |
702155 |
2.1.2.3 | -999 |
- |
N-([5-[2-(2,4-diaminoquinazolin-6-yl)ethyl]-2,3-dihydrothiophen-2-yl]carbonyl)-4-methylideneglutamic acid |
value above 0.05 |
702155 |
2.1.2.3 | -999 |
- |
N-[4-[2-(2,4-diamino-7H-pyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoyl]-4-methylideneglutamic acid |
value above 0.05 |
702155 |
2.1.2.3 | -999 |
- |
N-[4-[2-(2,4-diaminopyrido[3,2-d]pyrimidin-6-yl)ethyl]benzoyl]-4-methylideneglutamic acid |
value above 0.05 |
702155 |
2.1.2.3 | -999 |
- |
N-[4-[2-(2,4-diaminoquinazolin-6-yl)ethyl]-2-fluorobenzoyl]-4-methylideneglutamic acid |
value above 0.05 |
702155 |
2.1.2.3 | -999 |
- |
N-[4-[2-(2,4-diaminoquinazolin-6-yl)ethyl]benzoyl]-4-methylideneglutamic acid |
value above 0.05 |
702155 |
2.1.2.3 | -999 |
- |
N-[4-[2-(2-amino-4-methylquinazolin-6-yl)ethyl]benzoyl]-4-methylideneglutamic acid |
value above 0.05 |
702155 |
2.1.2.3 | 0.000005 |
- |
5-(5,5-dimethyl-6-oxo-1,4-dihydropyridin-3-yl)-N-(6-fluoro-1-oxo-2H-isoquinolin-7-yl)thiophene-2-sulfonamide |
IC50 below 0.000005 mM, at pH 7.5 and 25°C |
757394 |
2.1.2.3 | 0.000005 |
- |
5-(5-ethyl-5-methyl-6-oxo-1,4-dihydropyridin-3-yl)-N-(6-fluoro-1-oxo-2H-isoquinolin-7-yl)thiophene-2-sulfonamide |
IC50 below 0.000005 mM, at pH 7.5 and 25°C |
757394 |
2.1.2.3 | 0.000005 |
- |
N-(6-fluoro-1-oxo-2H-isoquinolin-7-yl)-5-(6-oxo-1H-pyridin-3-yl)thiophene-2-sulfonamide |
IC50 below 0.000005 mM, at pH 7.5 and 25°C |
757394 |