EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   1.4.1.3 | 0.00017 |
- |
GTP |
inhibition of wild-type enzyme and mutant enzymes r470H and N498S. No inhibition of mutant enzyme G456A. IC50 of mutant enzyme R470G is 0.00017 mM, IC50 of mutant enzyme N49 |
656060 |
| 1.4.1.3 | 0.00019 |
- |
GTP |
inhibition of wild-type enzyme and mutant enzymes r470H and N498S. No inhibition of mutant enzyme G456A. IC50 of wild-type enzyme is 0.00019 mM |
656060 |
| 1.4.1.3 | 0.00019 |
- |
GTP |
potent inhibitor. IC50 for wild-type enzyme is 0.00019 mM |
656871 |
| 1.4.1.3 | 0.00031 |
- |
GTP |
in the absence of other modulators, pH 8.0 |
700428 |
| 1.4.1.3 | 0.001 |
- |
corticosterone |
pH 8.0, temperature not specified in the publication |
743356 |
| 1.4.1.3 | 0.001 |
- |
diethylstilbestrol |
presence of 0.1 M ADP, pH 8.0, temperature not specified in the publication |
743356 |
| 1.4.1.3 | 0.001 |
- |
GTP |
isozyme GDH1 |
684905 |
| 1.4.1.3 | 0.0015 |
- |
17beta-estradiol |
pH 8.0, temperature not specified in the publication |
743356 |
| 1.4.1.3 | 0.00161 |
- |
GTP |
in the presence of 0.1 mM ADP, pH 8.0 |
700428 |
| 1.4.1.3 | 0.00167 |
- |
diethylstilbestrol |
pH 8.0, temperature not specified in the publication |
743356 |
