EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.2.1.104 | 0.0000026 |
- |
3-deazathiamine diphosphate |
pH 7.8, temperature not specified in the publication |
763321 |
1.2.1.104 | 0.000025 |
- |
Oxythiamine diphosphate |
pH 7.8, temperature not specified in the publication |
763321 |
1.2.1.104 | 0.00054 |
- |
N-(4-[(2E)-2-[(4-amino-2-methylpyrimidin-5-yl)methylidene]hydrazinecarbonyl]phenyl)-N'-phenylurea |
pH 6.4, 37°C |
758907 |
1.2.1.104 | 0.00062 |
- |
N-(4-[(2E)-2-[(4-amino-2-methylpyrimidin-5-yl)methylidene]hydrazinecarbonyl]phenyl)-4-bromobenzamide |
pH 6.4, 37°C |
758907 |
1.2.1.104 | 0.00066 |
- |
N-(3-[(2E)-2-[(4-amino-2-methylpyrimidin-5-yl)methylidene]hydrazinecarbonyl]phenyl)-4-bromobenzamide |
pH 6.4, 37°C |
758907 |
1.2.1.104 | 0.00148 |
- |
[1-[(4-amino-2-methylpyrimidin-5-yl)methyl]-5-iodo-4,5-dihydro-1H-1,2,3-triazol-4-yl]methyl 4-chlorobenzoate |
isolated E1 component, pH 7.2, 37°C |
758908 |
1.2.1.104 | 0.00161 |
- |
[1-[(4-amino-2-methylpyrimidin-5-yl)methyl]-5-iodo-4,5-dihydro-1H-1,2,3-triazol-4-yl]methyl 4-fluorobenzoate |
isolated E1 component, pH 7.2, 37°C |
758908 |
1.2.1.104 | 0.00169 |
- |
[1-[(4-amino-2-methylpyrimidin-5-yl)methyl]-5-iodo-4,5-dihydro-1H-1,2,3-triazol-4-yl]methyl 4-nitrobenzoate |
isolated E1 component, pH 7.2, 37°C |
758908 |
1.2.1.104 | 0.00179 |
- |
[1-[(4-amino-2-methylpyrimidin-5-yl)methyl]-5-iodo-4,5-dihydro-1H-1,2,3-triazol-4-yl]methyl 3-chlorobenzoate |
isolated E1 component, pH 7.2, 37°C |
758908 |
1.2.1.104 | 0.00191 |
- |
N-(3-[(2E)-2-[(4-amino-2-methylpyrimidin-5-yl)methylidene]hydrazinecarbonyl]phenyl)-4-fluorobenzamide |
pH 6.4, 37°C |
758907 |