EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   1.14.99.66 | 0.000022 |
- |
3-((1S,2R)-2-(cyclobutylamino)cyclopropyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzamide |
pH not specified in the publication, temperature not specified in the publication |
754904 |
| 1.14.99.66 | 0.000147 |
- |
4-([[(1S,2R)-2-phenylcyclopropyl]amino]ethyl)benzene-1-sulfonamide |
pH 8.5, 22°C |
753492 |
| 1.14.99.66 | 0.000153 |
- |
histone H3 |
pH 7.5, 25°C, recombinant enzyme |
744347 |
| 1.14.99.66 | 0.000154 |
- |
PCPA-Lys-4 H3-11 |
pH not specified in the publication, temperature not specified in the publication |
753006 |
| 1.14.99.66 | 0.00018 |
- |
PCPA-Orn-4 H3-11 |
pH not specified in the publication, temperature not specified in the publication |
753006 |
| 1.14.99.66 | 0.000195 |
- |
4-([[(1S,2R)-2-phenylcyclopropyl]amino]ethyl)benzamide |
pH 8.5, 22°C |
753492 |
| 1.14.99.66 | 0.0048 |
- |
histone H3-1-21 |
pH 7.5, 25°C |
744347 |
| 1.14.99.66 | 0.00484 |
- |
histone H3 1-21 peptide |
pH 7.5, 25°C, recombinant enzyme |
744347 |
| 1.14.99.66 | 0.283 |
- |
3-[(E)-2-[2-(5-fluoro-2-hydroxyphenyl)pyridin-4-yl]ethenyl]N'-hydroxybenzene-1-carboximidamide |
pH not specified in the publication, temperature not specified in the publication |
752967 |
