EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   1.14.13.39 | 0.00006 |
- |
6-chloro-4-(3-aminopropoxy)-1-benzopyran-2-one trifluoroacetic acid salt |
IC50: 60 nM, pharmacokinetic profile |
672524 |
| 1.14.13.39 | 0.00009 |
- |
6-chloro-4-(3-aminopropoxy)-1-benzopyran-2-one trifluoroacetic acid salt |
IC50: 90 nM, pharmacokinetic profile |
672524 |
| 1.14.13.39 | 0.00011 |
- |
6-chloro-4-(3-methylamino-propoxy)-1-benzopyran-2-one trifluoroacetic acid salt |
IC50: 0.00011mM |
672524 |
| 1.14.13.39 | 0.00025 |
- |
6-chloro-4-(3-methylamino-propoxy)-1-benzopyran-2-one trifluoroacetic acid salt |
IC50: 0.00025mM |
672524 |
| 1.14.13.39 | 0.00041 |
- |
4-(3-amino-propoxy)-6-chloro-1H-quinolin-2-one trifluoroacetic acid salt |
IC50: 410 nM, pharmacokinetic profile |
672524 |
| 1.14.13.39 | 0.00053 |
- |
6-chloro-4-(3-methylamino-propoxy)-1-benzopyran-2-one trifluoroacetic acid salt |
IC50: 0.00053mM |
672524 |
| 1.14.13.39 | 0.00056 |
- |
6-chloro-4-(3-aminopropoxy)-1-benzopyran-2-one trifluoroacetic acid salt |
IC50: 0.00056 mM, pharmacokinetic profile |
672524 |
| 1.14.13.39 | 0.0012 |
- |
6-chloro-4-(3-dimethylamino-propoxy)-1-benzopyran-2-one hydrochloric acid salt |
IC50: 0.0012 mM |
672524 |
| 1.14.13.39 | 0.0026 |
- |
4-(3-dimethylamino-propoxy)-1H-quinolin-2-one |
IC50: 0.0026 mM |
672524 |
| 1.14.13.39 | 0.0027 |
- |
7-nitroindazole |
pH 7.4, 35°C |
745312 |
