EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.14.11.65 | 0.000153 |
- |
histone H3 |
pH 7.5, 25°C, recombinant enzyme |
744347 |
1.14.11.65 | 0.0034 |
- |
7-[(5-aminopentyl)oxy]-N2-[3-(dimethylamino)propyl]-6-methoxy-N4,N4-dimethylquinazoline-2,4-diamine |
pH and temperature not specified in the publication |
757427 |
1.14.11.65 | 0.0037 |
- |
7-[(5-aminopentyl)oxy]-N4-(1-benzylpiperidin-4-yl)-N2-[3-(dimethylamino)propyl]-6-methoxyquinazoline-2,4-diamine |
pH and temperature not specified in the publication |
757427 |
1.14.11.65 | 0.00484 |
- |
H3 1-21 peptide |
pH 7.5, 25°C, recombinant enzyme |
744347 |
1.14.11.65 | 0.00484 |
- |
peptide H31-21 |
pH 7.5, 25°C |
744347 |
1.14.11.65 | 0.0165 |
- |
N-(1-benzylpiperidin-4-yl)-6,7-dimethoxy-2-(4-methyl-1,4-diazepan-1-yl)quinazolin-4-amine |
pH and temperature not specified in the publication |
757427 |
1.14.11.65 | 0.019 |
- |
7-[(5-aminopentyl)oxy]-6-methoxy-N2,N2,N4,N4-tetramethylquinazoline-2,4-diamine |
pH and temperature not specified in the publication |
757427 |
1.14.11.65 | 0.067 |
- |
N-oxalylglycine |
pH and temperature not specified in the publication |
745939 |