EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.1.1.95 | 0.00166 |
- |
ixocarpalactone A |
pH and temperature not specified in the publication |
763147 |
1.1.1.95 | 0.0025 |
- |
N-(4,6-dimethylpyridin-2-yl)-4-(4-(trifluoromethyl)benzyl)piperazine-1-carbothioamide |
pH and temperature not specified in the publication |
763147 |
1.1.1.95 | 0.0025 |
- |
N-(4,6-dimethylpyridin-2-yl)-4-[[4-(trifluoromethyl)phenyl]methyl]piperazine-1-carbothioamide |
pH 8.0, 22°C |
762795 |
1.1.1.95 | 0.0037 |
- |
N-(4,6-dimethylpyridin-2-yl)-4-[5-(trifluoromethyl)pyridin-2-yl]piperazine-1-carbothioamide |
pH 8.0, 22°C |
762795 |
1.1.1.95 | 0.0043 |
- |
N-(4,6-dimethylpyridin-2-yl)-4-[4-(trifluoromethyl)phenyl]piperazine-1-carbothioamide |
pH 8.0, 22°C |
762795 |
1.1.1.95 | 0.0053 |
- |
N-(4,6-dimethylpyridin-2-yl)-4-[[3-(trifluoromethyl)phenyl]methyl]piperazine-1-carbothioamide |
pH 8.0, 22°C |
762795 |
1.1.1.95 | 0.0057 |
- |
N-(4,6-dimethylpyridin-2-yl)-3-[4-(trifluoromethyl)anilino]piperidine-1-carbothioamide |
pH 8.0, 22°C |
762795 |
1.1.1.95 | 0.0058 |
- |
N-(4,6-dimethylpyridin-2-yl)-3-(hydroxymethyl)-4-[[4-(trifluoromethyl)phenyl]methyl]piperazine-1-carbothioamide |
pH 8.0, 22°C |
762795 |
1.1.1.95 | 0.0063 |
- |
N-(4,6-dimethylpyridin-2-yl)-4-[3-(trifluoromethyl)phenyl]piperazine-1-carbothioamide |
pH 8.0, 22°C |
762795 |
1.1.1.95 | 0.0063 |
- |
N-(4,6-dimethylpyridin-2-yl)-4-[[2-(trifluoromethyl)phenyl]methyl]piperazine-1-carbothioamide |
pH 8.0, 22°C |
762795 |