EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor  |
Reference |
|---|
    4.4.1.20 | 0.000135 |
- |
2-benzoyl-5-(5-[(4-chlorophenyl)(methyl)amino]pyridine-2-carbonyl)benzoic acid |
pH 7.8, temperature not specified in the publication, recombinant enzyme |
730788 |
| 4.4.1.20 | 0.000116 |
- |
2-benzoyl-5-[5-[(4-chlorophenyl)(methyl)amino]pyridine-2-carbonyl]benzoic acid |
pH not specified in the publication, temperature not specified in the publication |
748456 |
| 4.4.1.20 | 0.000095 |
- |
5-[5-[(4-chlorophenyl)(cyclopropylmethyl)amino]pyridine-2-carbonyl]-2-(4-methoxybenzoyl)benzoic acid |
pH not specified in the publication, temperature not specified in the publication |
748456 |
| 4.4.1.20 | 0.000017 |
- |
5-[5-[(4-chlorophenyl)(methyl)amino]pyridine-2-carbonyl]-2-(4-methoxybenzoyl)benzoic acid |
cell-free assay, the substrate LTA4 is produced in situ, 37°C, pH not specified in the publication |
747181 |
| 4.4.1.20 | 0.000124 |
- |
5-[5-[(4-chlorophenyl)(methyl)amino]pyridine-2-carbonyl]-2-(4-methoxybenzoyl)benzoic acid |
pH not specified in the publication, temperature not specified in the publication |
748456 |
| 4.4.1.20 | 0.05 |
- |
diethylcarbamazine |
IC50: 0.05 mM |
644493 |
| 4.4.1.20 | 1.9 |
- |
estrone-3-sulfate |
IC50: 1.9 mM |
644509 |
| 4.4.1.20 | 1.4 |
- |
hexylglutathione |
IC50: 1.4 mM |
644496 |
| 4.4.1.20 | 1 |
- |
indomethacin |
IC50: 1.0 mM |
644490 |
| 4.4.1.20 | 0.0011 |
- |
leukotriene C2 |
IC50: 0.0011 mM |
644504 |
