EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor  |
Reference |
|---|
   3.4.22.69 | 0.0042 |
- |
(-)-epigallocatechin-3-gallate |
pH not specified in the publication, temperature not specified in the publication |
764084 |
| 3.4.22.69 | 0.025 |
- |
(-)-epigallocatechin-3-gallate |
pH not specified in the publication, temperature not specified in the publication |
764084 |
| 3.4.22.69 | 0.0071 |
- |
(2E)-1-[3-(2-hydroperoxy-3-methylbut-3-en-1-yl)-2-hydroxy-4-methoxyphenyl]-3-(4-hydroxyphenyl)prop-2-en-1-one |
pH and temperature not specified in the publication |
753268 |
| 3.4.22.69 | 0.005 |
- |
(2E)-N-[2-[4-(dimethylamino)butyl]phenyl]-3-phenylprop-2-enamide |
pH and temperature not specified in the publication |
731443 |
| 3.4.22.69 | 0.44 |
- |
(2S)-2-(8[(1R,3S,4aR,8aS)-1-[[butyl(methyl)amino]methyl]octahydro-1H-2-benzopyran-3-yl]methyl]amino)-3-(1H-imidazol-4-yl)propanal |
pH 7.5, 37°C, mutant enzyme R188I |
752975 |
| 3.4.22.69 | 0.78 |
- |
(2S)-2-([(1R,3R,4aR,8aS)-1-8[butyl(methyl)amino]methyl]octahydro-1H-2-benzopyran-3-yl]methyl]amino)-3-(1H-imidazol-4-yl)propanal |
pH 7.5, 37°C, mutant enzyme R188I |
752975 |
| 3.4.22.69 | 0.26 |
- |
(2S)-2-([[(1S,3R,4aR,8aS)-1-[[butyl(methyl)amino]methyl]octahydro-1H-2-benzopyran-3-yl]methyl]amino)-3-(1H-imidazol-4-yl)propanal |
pH 7.5, 37°C, mutant enzyme R188I |
752975 |
| 3.4.22.69 | 0.095 |
- |
(2S)-2-([[(1S,3S,4aR,8aS)-1[butyl(methyl)amino]methyl]octahydro-1H-2-benzopyran-3-yl]methylamino)-3-(1H-imidazol-4-yl)propanal |
pH 7.5, 37°C, mutant enzyme R188I |
752975 |
| 3.4.22.69 | 0.42 |
- |
(2S)-2-([[(1S,4aR,8aS)-1-[[benzyl(methyl)amino]methyl]octahydro-1H-2-benzopyran-3-yl]methyl]amino)-3-(1H-imidazol-4-yl)propanal |
pH 7.5, 37°C, mutant enzyme R188I |
752975 |
| 3.4.22.69 | 0.1 |
- |
(2S)-2-([[(1S,4aR,8aS)-1-[[butyl(methyl)amino]methyl]octahydro-1H-2-benzopyran-3-yl]methyl]amino)-3-(1H-imidazol-4-yl)propanal |
pH 7.5, 37°C, mutant enzyme R188I |
752975 |
