EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.4.2.30 | 0.02 |
- |
suramin |
25°C, pH not specified in the publication |
722786 |
2.4.2.30 | 0.0858 |
- |
N-(acridin-9-yl)-4-nitrobenzamide |
25°C, pH not specified in the publication |
722786 |
2.4.2.30 | 0.086 |
- |
N-[2-oxo-4-(phenylamino)-3,8a-dihydro-2H-chromen-3-yl]acetamide |
25°C, pH not specified in the publication |
722786 |
2.4.2.30 | 0.157 |
- |
V8 protease |
25°C, pH not specified in the publication |
722786 |
2.4.2.30 | 0.019 |
- |
3-(4-oxo-3,5,6,7-tetrahydro-4H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-2-yl)propanoic acid |
at pH 7.5 and 22°C |
736518 |
2.4.2.30 | 0.0249 |
- |
4-(4-oxo-3,4-dihydroquinazolin-2-yl)butanoic acid |
at pH 7.5 and 22°C |
736518 |
2.4.2.30 | 0.0479 |
- |
3-(4-oxo-3,4,5,6,7,8-hexahydro[1]benzothieno[2,3-d]pyrimidin-2-yl)propanoic acid |
at pH 7.5 and 22°C |
736518 |
2.4.2.30 | 0.0524 |
- |
2-(3-hydroxypropyl)-3,5,6,7-tetrahydro-4H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-4-one |
at pH 7.5 and 22°C |
736518 |
2.4.2.30 | 0.135 |
- |
3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanoic acid |
at pH 7.5 and 22°C |
736518 |
2.4.2.30 | 0.169 |
- |
2-(3-hydroxypropyl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3H)-one |
at pH 7.5 and 22°C |
736518 |