EC Number   |
IC50 Value   |
IC50 Value Maximum   |
Inhibitor   |
Reference   |
|---|
 2.1.1.366 | 0.0008 |
- |
N2-[3'-[(4-[4-[3-(dimethylamino)propyl]piperazin-1-yl]pyridine-2-carbonyl)amino][1,1'-biphenyl]-4-carbonyl]-6-pyrrolidin-1-yl-L-norleucinamide |
pH and temperature not specified in the publication |
777166 |
 2.1.1.366 | 0.0012 |
- |
N2-[3'-[(4-[4-[3-(dimethylamino)propyl]piperazin-1-yl]pyridine-2-carbonyl)amino][1,1'-biphenyl]-4-carbonyl]-N6,N6-dimethyl-L-lysinamide |
pH and temperature not specified in the publication |
777166 |
 2.1.1.366 | 0.0023 |
- |
N-[[1,1'-bi(cyclohexan)]-4-yl]-6-methoxy-7-[3-(piperidin-1-yl)propoxy]-2-[4-(propan-2-yl)-1,4-diazepan-1-yl]quinazolin-4-amine |
pH and temperature not specified in the publication |
777166 |
 2.1.1.366 | 0.0031 |
- |
N2-(3'-[[4-(4-butylpiperazin-1-yl)pyridine-2-carbonyl]amino][1,1'-biphenyl]-4-carbonyl)-N6,N6-dimethyl-L-lysinamide |
pH and temperature not specified in the publication |
777166 |
 2.1.1.366 | 0.0032 |
- |
N2-(3'-[[4-(4-butylpiperazin-1-yl)pyridine-2-carbonyl]amino][1,1'-biphenyl]-4-carbonyl)-6-pyrrolidin-1-yl-L-norleucinamide |
pH and temperature not specified in the publication |
777166 |
 2.1.1.366 | 0.0034 |
- |
N4-[6-(dimethylamino)hexyl]-N2-[5-(dimethylamino)pentyl]-6,7-dimethoxyquinazoline-2,4-diamine |
pH and temperature not specified in the publication |
777166 |
 2.1.1.366 | 0.0035 |
- |
N2-(3'-[[4-(4-methylpiperazin-1-yl)pyridine-2-carbonyl]amino][1,1'-biphenyl]-4-carbonyl)-6-pyrrolidin-1-yl-L-norleucinamide |
pH and temperature not specified in the publication |
777166 |