EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.4.22.69 | 0.00003 |
- |
5-chloropyridin-3-yl 1H-indole-4-carboxylate |
pH and temperature not specified in the publication |
731443 |
| 3.4.22.69 | 0.000051 |
- |
2-(1H-benzotriazol-1-yl)-N-(biphenyl-4-yl)-N-(thiophen-3-ylmethyl)acetamide |
pH and temperature not specified in the publication |
731443 |
| 3.4.22.69 | 0.00006 |
- |
5-chloropyridin-3-yl 5-(4-nitrophenyl)-2-furoate |
- |
678619 |
| 3.4.22.69 | 0.00006 |
- |
N-(2-chloro-4-nitrophenyl)-Nalpha-[[4-(dimethylamino)phenyl]carbonyl]phenylalaninamide |
- |
679402 |
| 3.4.22.69 | 0.000063 |
- |
5-chloropyridin-3-yl 5-(4-chlorophenyl)-2-furoate |
- |
678619 |
| 3.4.22.69 | 0.000065 |
- |
(S)-N-((S)-1-(((S)-1-(1H-imidazol-4-yl)-3-oxopropan-2-yl)amino)-3-cyclohexyl-1-oxopropan-2-yl)-2-((S)-2-((S)-2-acetamido-3-hydroxypropanamido)propanamido)-3-methylbutanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
| 3.4.22.69 | 0.000065 |
- |
N-acetyl-Ser-Ala-Val-Cha-His |
in 10 mM Tris-HCl buffer, pH 7.5, containing 7 mM dithiothreitol, at 37°C |
717978 |
| 3.4.22.69 | 0.00008 |
- |
5-chloropyridin-3-yl 1H-indole-7-carboxylate |
- |
691304 |
| 3.4.22.69 | 0.000089 |
- |
5-chloropyridin-3-yl 1-[(3-nitrophenyl)sulfonyl]-1H-indole-5-carboxylate |
- |
691304 |
| 3.4.22.69 | 0.000108 |
- |
5-chloropyridin-3-yl 2-oxo-2H-chromene-3-carboxylate |
- |
678619 |
