EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.51 | 0.00004 |
- |
chloro[2,2'-(thio-kappaS)bis[ethanethiolato-kappaS]] oxorhenium(V) |
- |
699388 |
3.4.22.51 | 0.00007 |
- |
(2Z)-2-[1-(4-bromophenyl)-2-(3-chloro-4-fluorophenoxy)ethylidene]hydrazine-1-carbothioamide |
23°C, pH 5.5 |
753481 |
3.4.22.51 | 0.00007 |
- |
aceto[2,6-bis[(butylthio-jS)methyl]phenyl-kappaC]-,(SP-4-3)-palladium(II) |
- |
699388 |
3.4.22.51 | 0.00008 |
- |
(1E)-1-(3,4-dichlorophenyl)-2-phenylethan-1-one thiosemicarbazone |
IC50: 80 nM |
667951 |
3.4.22.51 | 0.0001 |
- |
Nalpha-[(2R,3E)-2-benzyl-4-(phenylsulfonyl)but-3-enoyl]-N-[(4-methylpiperazin-1-yl)carbonyl]-L-phenylalaninamide |
- |
696645 |
3.4.22.51 | 0.0002 |
- |
(3S,5R,11R)-N-benzyl-3-(2-methylpropyl)-2-oxo-11-[(E)-2-(phenylsulfonyl)ethenyl]-1,4-diazacycloundecane-5-carboxamide |
- |
696645 |
3.4.22.51 | 0.00031 |
- |
(1E)-1-(3-bromophenyl)propan-1-one thiosemicarbazone |
IC50: 310 nM |
667951 |
3.4.22.51 | 0.00035 |
- |
(p-methoxyphenylthiolato-S)[2,6-bis[(mercapto-kappaS)methyl]pyridine-kappaN] oxorhenium(V) |
- |
699388 |
3.4.22.51 | 0.0004 |
- |
(2Z)-2-[1-(4-bromophenyl)-2-(4-fluorophenoxy)ethylidene]hydrazine-1-carbothioamide |
23°C, pH 5.5 |
753481 |
3.4.22.51 | 0.0006 |
- |
(2E)-2-[1-([1,1'-biphenyl]-4-yl)-2-(4-bromophenoxy)ethylidene]hydrazine-1-carbothioamide |
23°C, pH 5.5 |
753481 |