EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.4.21.27 | 0.0773 |
- |
benzamidine |
- |
683239 |
| 3.4.21.27 | 0.1031 |
- |
N-[[5-chloro-2-(prop-2-en-1-yl)-1H-indol-3-yl]methyl]-N2-[(2R)-2-cyclohexyl-2-(pent-4-enoylamino)acetyl]-L-leucinamide |
pH and temperature not specified in the publication |
717333 |
| 3.4.21.27 | 0.12 |
- |
boronic acid |
- |
683239 |
| 3.4.21.27 | 0.1358 |
- |
(4S,7S,10S,12Z)-18-chloro-7-cyclohexyl-4-(2-methylpropyl)-10-phenyl-4,5,7,8,10,11,14,15-octahydro-1H-[1,4,7]triazacyclohexadecino[10,9-b]indole-3,6,9(2H)-trione |
pH and temperature not specified in the publication |
717333 |
| 3.4.21.27 | 0.1459 |
- |
N-[[5-chloro-2-(prop-2-en-1-yl)-1H-indol-3-yl]methyl]-N2-[(2R)-2-cyclohexyl-2-[[(2S)-2-phenylpent-4-enoyl]amino]acetyl]-L-leucinamide |
pH and temperature not specified in the publication |
717333 |
| 3.4.21.27 | 0.1759 |
- |
(4S,7S)-18-chloro-7-cyclohexyl-4-(2-methylpropyl)-1,2,4,5,7,8,10,11,12,13,14,15-dodecahydro[1,2,5,8]thiatriazacyclohexadecino[11,10-b]indole-3,6-dione 9,9-dioxide |
pH and temperature not specified in the publication |
717333 |
| 3.4.21.27 | 0.7678 |
- |
(4S,7S,12Z)-18-chloro-7-cyclohexyl-4-(2-methylpropyl)-1,2,4,5,7,8,10,11,14,15-decahydro[1,2,5,8]thiatriazacyclohexadecino[11,10-b]indole-3,6-dione 9,9-dioxide |
pH and temperature not specified in the publication |
717333 |
